Exploiting an Asp-Glu "switch" in glycogen synthase kinase 3 to design paralog-selective inhibitors for use in acute myeloid leukemia
利用糖原合酶激酶 3 中的 Asp-Glu“开关”设计用于治疗急性髓系白血病的同源物选择性抑制剂
期刊:Science Translational Medicine
影响因子:15.8
doi:10.1126/scitranslmed.aam8460
Florence F Wagner, Lina Benajiba, Arthur J Campbell, Michel Weïwer, Joshua R Sacher, Jennifer P Gale, Linda Ross, Alexandre Puissant, Gabriela Alexe, Amy Conway, Morgan Back, Yana Pikman, Ilene Galinsky, Daniel J DeAngelo, Richard M Stone, Taner Kaya, Xi Shi, Matthew B Robers, Thomas Machleidt, Jenn