日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications

立体选择性和区域选择性明确的DNA编码化学库能够实现高效的肿瘤靶向应用

Favalli, Nicholas; Bassi, Gabriele; Pellegrino, Christian; Millul, Jacopo; De Luca, Roberto; Cazzamalli, Samuele; Yang, Su; Trenner, Anika; Mozaffari, Nour L; Myburgh, Renier; Moroglu, Mustafa; Conway, Stuart J; Sartori, Alessandro A; Manz, Markus G; Lerner, Richard A; Vogt, Peter K; Scheuermann, Jörg; Neri, Dario

Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain

在设计 CREBBP 溴结构域的选择性高亲和力配体时控制分子内相互作用

Michael Brand, James Clayton, Mustafa Moroglu, Matthias Schiedel, Sarah Picaud, Joseph P Bluck, Anna Skwarska, Hannah Bolland, Anthony K N Chan, Corentine M C Laurin, Amy R Scorah, Larissa See, Timothy P C Rooney, Katrina H Andrews, Oleg Fedorov, Gabriella Perell, Prakriti Kalra, Kayla B Vinh, Wilia

A Single-Stranded DNA-Encoded Chemical Library Based on a Stereoisomeric Scaffold Enables Ligand Discovery by Modular Assembly of Building Blocks

基于立体异构骨架的单链DNA编码化学库可通过模块化组装构建模块实现配体发现

Bassi, Gabriele; Favalli, Nicholas; Vuk, Miriam; Catalano, Marco; Martinelli, Adriano; Trenner, Anika; Porro, Antonio; Yang, Su; Tham, Chuin Lean; Moroglu, Mustafa; Yue, Wyatt W; Conway, Stuart J; Vogt, Peter K; Sartori, Alessandro A; Scheuermann, Jörg; Neri, Dario

BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability

BET 溴结构域配体:探索 WPF 架以提高 BRD4 溴结构域亲和力和代谢稳定性

Laura E Jennings, Matthias Schiedel, David S Hewings, Sarah Picaud, Corentine M C Laurin, Paul A Bruno, Joseph P Bluck, Amy R Scorah, Larissa See, Jessica K Reynolds, Mustafa Moroglu, Ishna N Mistry, Amy Hicks, Pavel Guzanov, James Clayton, Charles N G Evans, Giulia Stazi, Philip C Biggin, Anna K Ma

Seroprevalence of Hepatitis A Virus Antibodies among the Patients with Chronic Hepatitis B in Turkey

土耳其慢性乙型肝炎患者中甲型肝炎病毒抗体的血清阳性率

Tulek, Necla; Ozsoy, Metin; Moroglu, Cigdem; Cagla Sonmezer, Meliha; Temocin, Fatih; Tuncer Ertem, Gunay; Sebnem Erdinc, Fatma

Giant intraoral condyloma accuminatum lesion coexisting with genital condyloma

巨大口腔内尖锐湿疣病变与生殖器尖锐湿疣并存

Ozdamar, S Serap Moroglu; Ozdamar, Ozkan; Kucukodaci, Zafer

Indirect measurement of the temporomandibular joint disc elasticity with magnetic resonance imaging

利用磁共振成像间接测量颞下颌关节盘弹性

Yildirim, D; Dergin, G; Tamam, C; Moroglu, S; Gurses, B