Development and Pharmacochemical Characterization Discover a Novel Brain-Permeable HDAC11-Selective Inhibitor with Therapeutic Potential by Regulating Neuroinflammation in Mice
开发和药理化学表征:发现一种新型的可穿透血脑屏障的HDAC11选择性抑制剂,该抑制剂可通过调节小鼠神经炎症发挥治疗潜力
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.3c01491
Bai, Ping; Liu, Yan; Yang, Liuyue; Ding, Weihua; Mondal, Prasenjit; Sang, Na; Liu, Gang; Lu, Xiaoxia; Ho, Thanh Tu; Zhou, Yanting; Wu, Rui; Birar, Vishal C; Wilks, Moses Q; Tanzi, Rudolph E; Lin, Hening; Zhang, Can; Li, Weimin; Shen, Shiqian; Wang, Changning