日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Neobavaisoflavone Induces Bilirubin Metabolizing Enzyme UGT1A1 via PPARα and PPARγ

新巴伐利亚异黄酮通过 PPARα 和 PPARγ 诱导胆红素代谢酶 UGT1A1

Ya-Di Zhu, Xiao-Qing Guan, Jing Chen, Sheng Peng, Moshe Finel, Ying-Yuan Zhao, Rui-Min Wang, Hui-Chang Bi, Ming Lei, Dan-Dan Wang, Guang-Bo Ge

An ultra-sensitive and easy-to-use assay for sensing human UGT1A1 activities in biological systems

一种超灵敏且易于使用的检测方法,用于检测生物系统中人类 UGT1A1 的活性

Ya-Di Zhu, Hui-Lin Pang, Qi-Hang Zhou, Zi-Fei Qin, Qiang Jin, Moshe Finel, Yi-Nan Wang, Wei-Wei Qin, Yin Lu, Dan-Dan Wang, Guang-Bo Ge

Molecular Docking-Based Design and Development of a Highly Selective Probe Substrate for UDP-glucuronosyltransferase 1A10

基于分子对接的 UDP-葡萄糖醛酸转移酶 1A10 高选择性探针底物的设计和开发

Risto O Juvonen, Sanna Rauhamäki, Sami Kortet, Sanna Niinivehmas, Johanna Troberg, Aleksanteri Petsalo, Juhani Huuskonen, Hannu Raunio, Moshe Finel, Olli T Pentikäinen

Albumin stimulates the activity of the human UDP-glucuronosyltransferases 1A7, 1A8, 1A10, 2A1 and 2B15, but the effects are enzyme and substrate dependent

白蛋白可刺激人类 UDP-葡萄糖醛酸转移酶 1A7、1A8、1A10、2A1 和 2B15 的活性,但其作用依赖于酶和底物

Nenad Manevski, Johanna Troberg, Paolo Svaluto-Moreolo, Klaudyna Dziedzic, Jari Yli-Kauhaluoma, Moshe Finel

Role of human UDP-glucuronosyltransferases in the biotransformation of the triazoloacridinone and imidazoacridinone antitumor agents C-1305 and C-1311: highly selective substrates for UGT1A10

人类 UDP-葡萄糖醛酸转移酶在三唑并吖啶酮和咪唑并吖啶酮抗肿瘤药物 C-1305 和 C-1311 的生物转化中的作用:UGT1A10 的高选择性底物

Barbara Fedejko-Kap, Stacie M Bratton, Moshe Finel, Anna Radominska-Pandya, Zofia Mazerska

Analysis of R- and S-hydroxywarfarin glucuronidation catalyzed by human liver microsomes and recombinant UDP-glucuronosyltransferases

人肝微粒体和重组UDP-葡萄糖醛酸转移酶催化的R-和S-羟基华法林葡萄糖醛酸化分析

Stacie M Bratton, Carrie M Mosher, Farid Khallouki, Moshe Finel, Michael H Court, Jeffery H Moran, Anna Radominska-Pandya

Glucuronidation of psilocin and 4-hydroxyindole by the human UDP-glucuronosyltransferases

人类 UDP-葡萄糖醛酸转移酶对裸盖菇素和 4-羟基吲哚进行葡萄糖醛酸化

Nenad Manevski, Mika Kurkela, Camilla Höglund, Timo Mauriala, Michael H Court, Jari Yli-Kauhaluoma, Moshe Finel

Human UDP-glucuronosyltransferase UGT2A2: cDNA construction, expression, and functional characterization in comparison with UGT2A1 and UGT2A3

人类 UDP-葡萄糖醛酸转移酶 UGT2A2:与 UGT2A1 和 UGT2A3 相比的 cDNA 构建、表达和功能特征

Nina Sneitz, Michael H Court, Xiuling Zhang, Kaisa Laajanen, Karen K Yee, Pamela Dalton, Xinxin Ding, Moshe Finel