Identification of imidazo[1,2-b]pyridazine TYK2 pseudokinase ligands as potent and selective allosteric inhibitors of TYK2 signalling
鉴定咪唑并[1,2-b]哒嗪类TYK2假激酶配体为TYK2信号传导的强效选择性变构抑制剂
期刊:Medchemcomm
影响因子:
doi:10.1039/c6md00560h
Moslin, R; Gardner, D; Santella, J; Zhang, Y; Duncia, J V; Liu, C; Lin, J; Tokarski, J S; Strnad, J; Pedicord, D; Chen, J; Blat, Y; Zupa-Fernandez, A; Cheng, L; Sun, H; Chaudhry, C; Huang, C; D'Arienzo, C; Sack, J S; Muckelbauer, J K; Chang, C; Tredup, J; Xie, D; Aranibar, N; Burke, J R; Carter, P H; Weinstein, D S