日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Simulating Intestinal Transporter and Enzyme Activity in a Physiologically Based Pharmacokinetic Model for Tenofovir Disoproxil Fumarate

在基于生理的药代动力学模型中模拟富马酸替诺福韦二吡呋酯的肠道转运体和酶活性

Moss, Darren M; Domanico, Paul; Watkins, Melynda; Park, Seonghee; Randolph, Ryan; Wring, Steve; Rajoli, Rajith Kumar Reddy; Hobson, James; Rannard, Steve; Siccardi, Marco; Owen, Andrew

Efavirenz Is Predicted To Accumulate in Brain Tissue: an In Silico, In Vitro, and In Vivo Investigation

依非韦伦预计会在脑组织中蓄积:一项计算机模拟、体外和体内研究

Curley, Paul; Rajoli, Rajith K R; Moss, Darren M; Liptrott, Neill J; Letendre, Scott; Owen, Andrew; Siccardi, Marco

Rilpivirine inhibits drug transporters ABCB1, SLC22A1, and SLC22A2 in vitro

利匹韦林在体外抑制药物转运蛋白ABCB1、SLC22A1和SLC22A2

Moss, Darren M; Liptrott, Neill J; Curley, Paul; Siccardi, Marco; Back, David J; Owen, Andrew

Divalent metals and pH alter raltegravir disposition in vitro.

二价金属和 pH 值会改变拉替拉韦在体外的处置

Moss Darren M, Siccardi Marco, Murphy Matthew, Piperakis Michael M, Khoo Saye H, Back David J, Owen Andrew