日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Deconstruction of Dual-Site Tankyrase Inhibitors Provides Insights into Binding Energetics and Suggests Critical Hotspots for Ligand Optimization.

双位点坦克酶抑制剂的解构为结合能学提供了见解,并提出了配体优化的关键热点

Sowa Sven T, Kücükdisli Murat, Mostinski Yelena, Schaller David A, Vinagreiro Carolina S, Cirillo Davide, Bosetti Chiara, Brinch Shoshy Alam, van Laar Kirsten, Wegert Anita, Leenders Ruben G G, Krauss Stefan, Waaler Jo, Volkamer Andrea, Lehtiö Lari, Nazaré Marc

Visualization of membrane localization and the functional state of CB(2)R pools using matched agonist and inverse agonist probe pairs

利用匹配的激动剂和反向激动剂探针对,可视化CB(2)R池的膜定位和功能状态。

Wąsińska-Kałwa, M; Omran, A; Mach, L; Scipioni, L; Bouma, J; Li, X; Radetzki, S; Mostinski, Y; Schippers, M; Gazzi, T; van der Horst, C; Brennecke, B; Hanske, A; Kolomeets, Y; Guba, W; Sykes, D; von Kries, J P; Broichhagen, J; Hua, T; Veprintsev, D; Heitman, L H; Oddi, S; Maccarrone, M; Grether, U; Nazare, M

Highly Selective Drug-Derived Fluorescent Probes for the Cannabinoid Receptor Type 1 (CB1R)

针对大麻素受体 1 型 (CB1R) 的高选择性药物衍生荧光探针

Leonard Mach, Anahid Omran, Jara Bouma, Silke Radetzki, David A Sykes, Wolfgang Guba, Xiaoting Li, Calvin Höffelmeyer, Axel Hentsch, Thais Gazzi, Yelena Mostinski, Malgorzata Wasinska-Kalwa, Fabio de Molnier, Cas van der Horst, Jens Peter von Kries, Marc Vendrell, Tian Hua, Dmitry B Veprintsev, Laur

Bacterial Colonization and Proliferation in Primary Molars following the Use of the Hall Technique: A Confocal Laser Scanning Microscopy Study

使用霍尔技术后乳磨牙中细菌定植和增殖情况:一项共聚焦激光扫描显微镜研究

Elbahary, Shlomo; Aharonian, Shiran; Azem, Hanaa; Peretz, Benjamin; Mostinski, Olga; Blumer, Sigalit

Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe

利用高效、细胞渗透性荧光探针检测天然细胞和斑马鱼中的大麻素受体2型

Gazzi, Thais; Brennecke, Benjamin; Atz, Kenneth; Korn, Claudia; Sykes, David; Forn-Cuni, Gabriel; Pfaff, Patrick; Sarott, Roman C; Westphal, Matthias V; Mostinski, Yelena; Mach, Leonard; Wasinska-Kalwa, Malgorzata; Weise, Marie; Hoare, Bradley L; Miljuš, Tamara; Mexi, Maira; Roth, Nicolas; Koers, Eline J; Guba, Wolfgang; Alker, André; Rufer, Arne C; Kusznir, Eric A; Huber, Sylwia; Raposo, Catarina; Zirwes, Elisabeth A; Osterwald, Anja; Pavlovic, Anto; Moes, Svenja; Beck, Jennifer; Nettekoven, Matthias; Benito-Cuesta, Irene; Grande, Teresa; Drawnel, Faye; Widmer, Gabriella; Holzer, Daniela; van der Wel, Tom; Mandhair, Harpreet; Honer, Michael; Fingerle, Jürgen; Scheffel, Jörg; Broichhagen, Johannes; Gawrisch, Klaus; Romero, Julián; Hillard, Cecilia J; Varga, Zoltan V; van der Stelt, Mario; Pacher, Pal; Gertsch, Jürg; Ullmer, Christoph; McCormick, Peter J; Oddi, Sergio; Spaink, Herman P; Maccarrone, Mauro; Veprintsev, Dmitry B; Carreira, Erick M; Grether, Uwe; Nazaré, Marc