日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Deconstruction of Dual-Site Tankyrase Inhibitors Provides Insights into Binding Energetics and Suggests Critical Hotspots for Ligand Optimization.

双位点坦克酶抑制剂的解构为结合能学提供了见解,并提出了配体优化的关键热点

Sowa Sven T, Kücükdisli Murat, Mostinski Yelena, Schaller David A, Vinagreiro Carolina S, Cirillo Davide, Bosetti Chiara, Brinch Shoshy Alam, van Laar Kirsten, Wegert Anita, Leenders Ruben G G, Krauss Stefan, Waaler Jo, Volkamer Andrea, Lehtiö Lari, Nazaré Marc

Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe

利用高效、细胞渗透性荧光探针检测天然细胞和斑马鱼中的大麻素受体2型

Gazzi, Thais; Brennecke, Benjamin; Atz, Kenneth; Korn, Claudia; Sykes, David; Forn-Cuni, Gabriel; Pfaff, Patrick; Sarott, Roman C; Westphal, Matthias V; Mostinski, Yelena; Mach, Leonard; Wasinska-Kalwa, Malgorzata; Weise, Marie; Hoare, Bradley L; Miljuš, Tamara; Mexi, Maira; Roth, Nicolas; Koers, Eline J; Guba, Wolfgang; Alker, André; Rufer, Arne C; Kusznir, Eric A; Huber, Sylwia; Raposo, Catarina; Zirwes, Elisabeth A; Osterwald, Anja; Pavlovic, Anto; Moes, Svenja; Beck, Jennifer; Nettekoven, Matthias; Benito-Cuesta, Irene; Grande, Teresa; Drawnel, Faye; Widmer, Gabriella; Holzer, Daniela; van der Wel, Tom; Mandhair, Harpreet; Honer, Michael; Fingerle, Jürgen; Scheffel, Jörg; Broichhagen, Johannes; Gawrisch, Klaus; Romero, Julián; Hillard, Cecilia J; Varga, Zoltan V; van der Stelt, Mario; Pacher, Pal; Gertsch, Jürg; Ullmer, Christoph; McCormick, Peter J; Oddi, Sergio; Spaink, Herman P; Maccarrone, Mauro; Veprintsev, Dmitry B; Carreira, Erick M; Grether, Uwe; Nazaré, Marc