日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of small molecules that enhance aminoglycoside-mediated suppression of CFTR and NF1 nonsense mutations.

鉴定能增强氨基糖苷类药物对 CFTR 和 NF1 无义突变抑制作用的小分子。

Sammons Joshua, Chen Jianguo, Thrasher Kari, Fu Lianwu, Du Ming, Wen Hui, Bostwick J Robert, Vinson Paige, Moukha-Chafiq Omar, Augelli-Szafran Corinne, Keeling Kim M, Wallis Deeann, Kesterson Robert A, Rowe Steven M, Bedwell David M

High-throughput screening for identification of influenza a inhibitors using a cell-based immunofluorescence assay.

利用基于细胞的免疫荧光检测方法进行高通量筛选,以鉴定甲型流感病毒抑制剂

Martinez-Gzegozewska Yohanka, Rasmussen Lynn, Nebane N Miranda, McKellip Sara, Radzieta Dee, Manuvakhova Anna, Reece Andrew J, Ruiz Pedro, Zhang Sixue, Moukha-Chafiq Omar, Sosa Melinda, Augelli-Szafran Corinne, Whitley Richard, Bostwick Robert, Vinson Paige

Synthesis and evaluation of novel substituted N-(2-phenylbutyl)-5,6,7,8-tetrahydro-quinazolin-4-amines as allosteric modulators of HIV-DAT-tat interaction

合成并评价新型取代的N-(2-苯基丁基)-5,6,7,8-四氢喹唑啉-4-胺作为HIV-DAT-tat相互作用的变构调节剂

Nguyen, Theresa H; Moukha-Chafiq, Omar; Karyakarte, Shuklendu; Jimenez-Torres, Ana C; Shrestha, Ganesh; Zhang, Sixue; Zhu, Jun; Augelli-Szafran, Corinne E

Development of Delta Opioid Receptor Antagonists Which Prevent Alzheimer's Disease-Like Pathology in the 5X-Familial Alzheimer's Disease [5XFAD] Mouse Model

开发δ阿片受体拮抗剂以预防5X家族性阿尔茨海默病[5XFAD]小鼠模型中阿尔茨海默病样病理的发生

Tanguturi, Parthasaradhireddy; Mitchell, Stefanie; Moukha-Chafiq, Omar; Zhang, Sixue; Tillotson, John; Ananthan, Subramaniam; Augelli-Szafran, Corinne E; Streicher, John M

Effects of SRI-32743, a Novel Quinazoline Structure-Based Compound, on HIV-1 Tat and Cocaine Interaction with Norepinephrine Transporter

新型喹唑啉结构化合物SRI-32743对HIV-1 Tat蛋白及可卡因与去甲肾上腺素转运蛋白相互作用的影响

Jiménez-Torres, Ana Catya; Porter, Katherine D; Hastie, Jamison A; Adeniran, Charles; Moukha-Chafiq, Omar; Nguyen, Theresa H; Ananthan, Subramaniam; Augelli-Szafran, Corinne E; Zhan, Chang-Guo; Zhu, Jun

The D3 receptor antagonist SR 21502 reduces cue-induced reinstatement of methamphetamine-seeking in rats

D3受体拮抗剂SR 21502可降低大鼠对甲基苯丙胺的线索诱导性复吸行为。

Ranaldi, Robert; Timken, Patrick; Parasram, Daleya; Ali, Tasmia; Zhang, Sixue; Moukha-Chafiq, Omar; Augelli-Szafran, Corinne; Streicher, John M

Correction: Tanguturi et al. Discovery of Novel Delta Opioid Receptor (DOR) Inverse Agonist and Irreversible (Non-Competitive) Antagonists. Molecules 2021, 26, 6693

更正:Tanguturi 等人,《新型δ阿片受体(DOR)反向激动剂和不可逆(非竞争性)拮抗剂的发现》,Molecules 2021, 26, 6693

Tanguturi, Parthasaradhireddy; Pathak, Vibha; Zhang, Sixue; Moukha-Chafiq, Omar; Augelli-Szafran, Corinne E; Streicher, John M

Inhibitors of HIV-1 Nef-Mediated Activation of the Myeloid Src-Family Kinase Hck Block HIV-1 Replication in Macrophages and Disrupt MHC-I Downregulation

HIV-1 Nef介导的髓系Src家族激酶Hck激活抑制剂可阻断巨噬细胞中的HIV-1复制并破坏MHC-I下调

Lori A Emert-Sedlak ,Omar Moukha-Chafiq, Haibin Shi ,Shoucheng Du ,John J Alvarado ,Vibha Pathak, Samuel G Tanner, Robert N Hunter, Miranda Nebane, Li Chen ,Tatiana V Ilina ,Rieko Ishima ,Sixue Zhang, Yury V Kuzmichev ,Elizabeth R Wonderlich ,Susan M Schader ,Corinne E Augelli-Szafran, Roger G Ptak ,Thomas E Smithgall

Design, Synthesis, and Antiprotozoal Evaluation of New Promising 2,9-Bis[(substituted-aminomethyl)]-4,7-phenyl-1,10-phenanthroline Derivatives, a Potential Alternative Scaffold to Drug Efflux

新型有前景的2,9-双[(取代氨甲基)]-4,7-苯基-1,10-菲咯啉衍生物的设计、合成及抗原生动物活性评价,一种潜在的药物外排替代骨架

Guillon, Jean; Cohen, Anita; Boudot, Clotilde; Monic, Sarah; Savrimoutou, Solène; Moreau, Stéphane; Albenque-Rubio, Sandra; Lafon-Schmaltz, Camille; Dassonville-Klimpt, Alexandra; Mergny, Jean-Louis; Ronga, Luisa; Bernabeu de Maria, Mikel; Lamarche, Jeremy; Lago, Cristina Dal; Largy, Eric; Gabelica, Valérie; Moukha, Serge; Dozolme, Pascale; Agnamey, Patrice; Azas, Nadine; Mullié, Catherine; Courtioux, Bertrand; Sonnet, Pascal

Targeting Chikungunya Virus Replication by Benzoannulene Inhibitors

利用苯并环烯类抑制剂靶向抑制基孔肯雅病毒复制

Ahmed, S Kaleem; Haese, Nicole N; Cowan, Jaden T; Pathak, Vibha; Moukha-Chafiq, Omar; Smith, Valerie J; Rodzinak, Kevin J; Ahmad, Fahim; Zhang, Sixue; Bonin, Kiley M; Streblow, Aaron D; Streblow, Cassilyn E; Kreklywich, Craig N; Morrison, Clayton; Sarkar, Sanjay; Moorman, Nathaniel; Sander, Wes; Allen, Robbie; DeFilippis, Victor; Tekwani, Babu L; Wu, Mousheng; Hirsch, Alec J; Smith, Jessica L; Tower, Nichole A; Rasmussen, Lynn; Bostwick, Robert; Maddry, Joseph A; Ananthan, Subramaniam; Gerdes, John M; Augelli-Szafran, Corinne E; Suto, Mark J; Morrison, Thomas E; Heise, Mark T; Streblow, Daniel N; Pathak, Ashish K