日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of [1,2,4]triazolo[1,5-a]pyrimidine-Imatinib Hybrids With Selective Cytotoxic Activity: A Mechanistically Divergent Series From Direct BCR-ABL1 Inhibition

发现具有选择性细胞毒活性的[1,2,4]三唑并[1,5-a]嘧啶-伊马替尼杂合物:与直接抑制BCR-ABL1机制不同的系列

Moura, Stefany Castro Bazan; de Oliveira, Andressa Paula; Neto, Joao de Mello Rezende; Dantas, Rafael Ferreira; Silva-Jr, Floriano Paes; Pimentel, Luiz Claudio; Carvalho, Mayara Salles do Nascimento; Leite, Debora Inacio; da Silva, Daiane Vitoria; Bastos, Monica Macedo; Boechat, Nubia

A Review on Medicinal Chemistry and Biological Activity of Dihydropyrimidinones Against HIV

二氢嘧啶酮类药物的药物化学及抗HIV生物活性研究综述

Leite, Debora I; Macedo, Fernando B; Lima, Murilo Marinho de C; Brum, Isabelle S; Oliveira, Jonathan Fragoso Miranda de; Costa, Ana Clara S; Duarte, Stella C; Moon, Sarah; Moura, Stefany de Castro B; Oliveira, Andressa P de; Boechat, Nubia; Bastos, Monica M

Ponatinib: A Review of the History of Medicinal Chemistry behind Its Development

帕纳替尼:其研发背后的药物化学史回顾

Nascimento, Mayara; Moura, Stefany; Parra, Lidia; Vasconcellos, Valeska; Costa, Gabriela; Leite, Debora; Dias, Maria; Fernandes, Tácio Vinício Amorim; Hoelz, Lucas; Pimentel, Luiz; Bastos, Monica; Boechat, Nubia

The transcriptional regulator Fur modulates the expression of uge, a gene essential for the core lipopolysaccharide biosynthesis in Klebsiella pneumoniae

转录调控因子Fur调节uge基因的表达,uge基因是肺炎克雷伯菌核心脂多糖生物合成所必需的基因。

Muner, José Júlio; de Oliveira, Paloma Aparecida Alves; Baboghlian, Juliana; Moura, Stefany Casarin; de Andrade, Abissair Gabriel; de Oliveira, Michelly Macedo; Campos, Yasmin Ferreira de; Mançano, Alquiandra Stefani Ferreira; Siqueira, Nathália Maria Gonçalves; Pacheco, Thaisy; Ferraz, Lúcio Fábio Caldas

A Review of the Development of Multitarget Molecules against HIV-TB Coinfection Pathogens

针对HIV-TB合并感染病原体的多靶点分子研发进展综述

Leite, Debora Inacio; de Castro Bazan Moura, Stefany; da Conceição Avelino Dias, Maria; Costa, Carolina Catta Preta; Machado, Gustavo Peixoto; Pimentel, Luiz Claudio Ferreira; Branco, Frederico Silva Castelo; Moreira, Rui; Bastos, Monica Macedo; Boechat, Nubia

New Imatinib Derivatives with Antiproliferative Activity against A549 and K562 Cancer Cells.

具有抗A549和K562癌细胞增殖活性的新型伊马替尼衍生物

Oliveira Andressa, Moura Stefany, Pimentel Luiz, Neto João, Dantas Rafael, Silva-Jr Floriano, Bastos Monica, Boechat Nubia