日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Nivolumab plus ipilimumab induce hyper-progression in renal medullary carcinoma: results of a phase II trial and preclinical evidence.

纳武利尤单抗联合伊匹木单抗可诱导肾髓质癌超进展:II期试验结果和临床前证据。

Soeung Melinda, Yan Xinmiao, Zanca Ciro, Qian Jing, Karki Menuka, Duan Fei, Khan Hania, Zhang Li, Peng David H, Williams Mariah, He Rong, Chen Ziheng, Perelli Luigi, Chen Jianfeng, Tidwell Rebecca S, Chauhan Pankaj K, Le Courtney N, Lam Truong N A, Bhattacharya Nirjar, Shah Rutvi, Ho I-Lin, Gay Jason P, Carrillo Caroline C, Feng Ningping, Le Kang, Gao Guang, Perry Teresa L, Mseeh Faika, Jiang Yongying, Xu Quanyun A, Zacharias Niki Marie, Sheth Rahul A, Bathala Tharakeswara K, Rao Priya, Daw Najat C, Tripathi Durga N, Walker Cheryl L, Mohammad Mohammad M, Zhang Jianhua, Han Guangchun, Chu Yanshuo, Wang Ruiping, Dang Minghao, Dai Enyu, Peng Fuduan, Liu Yunhe, Jadhav Akshaya, Lang Wenhua, Arrechedera Claudio A, Clemente Leticia Campos, Parra Edwin R, Lu Hsinyi, Haymaker Cara L, Wistuba Ignacio I, Futreal Andrew, Viale Andrea, Soth Michael J, Jones Philip, Marszalek Joseph R, Heffernan Timothy, Draetta Giulio F, Tannir Nizar M, Gao Jianjun, Wang Linghua, Genovese Giannicola, Msaouel Pavlos

Inhibition of dual leucine zipper kinase prevents chemotherapy-induced peripheral neuropathy and cognitive impairments

抑制双亮氨酸拉链激酶可预防化疗引起的周围神经病变和认知障碍

Jiacheng Ma, Sunil Goodwani, Paul J Acton, Virginie Buggia-Prevot, Shelli R Kesler, Imran Jamal, Iteeben D Mahant, Zhen Liu, Faika Mseeh, Bruce L Roth, Chaitali Chakraborty, Bo Peng, Qi Wu, Yongying Jiang, Kang Le, Michael J Soth, Philip Jones, Annemieke Kavelaars, William J Ray, Cobi J Heijnen

A Role for Protease Activated Receptor Type 3 (PAR3) in Nociception Demonstrated Through Development of a Novel Peptide Agonist

通过开发新型肽激动剂证明蛋白酶激活受体 3 型 (PAR3) 在伤害感受中的作用

Juliet Mwirigi, Moeno Kume, Shayne N Hassler, Ayesha Ahmad, Pradipta R Ray, Changyu Jiang, Alexander Chamessian, Nakleh Mseeh, Breya P Ludwig, Benjamin D Rivera, Marvin T Nieman, Thomas Van de Ven, Ru-Rong Ji, Gregory Dussor, Scott Boitano, Josef Vagner, Theodore J Price

Allosteric SHP2 Inhibitor, IACS-13909, Overcomes EGFR-Dependent and EGFR-Independent Resistance Mechanisms toward Osimertinib

变构SHP2抑制剂IACS-13909可克服EGFR依赖性和EGFR非依赖性奥希替尼耐药机制

Sun, Yuting; Meyers, Brooke A; Czako, Barbara; Leonard, Paul; Mseeh, Faika; Harris, Angela L; Wu, Qi; Johnson, Sarah; Parker, Connor A; Cross, Jason B; Di Francesco, Maria Emilia; Bivona, Benjamin J; Bristow, Christopher A; Burke, Jason P; Carrillo, Caroline C; Carroll, Christopher L; Chang, Qing; Feng, Ningping; Gao, Guang; Gera, Sonal; Giuliani, Virginia; Huang, Justin K; Jiang, Yongying; Kang, Zhijun; Kovacs, Jeffrey J; Liu, Chiu-Yi; Lopez, Anastasia M; Ma, Xiaoyan; Mandal, Pijus K; McAfoos, Timothy; Miller, Meredith A; Mullinax, Robert A; Peoples, Michael; Ramamoorthy, Vandhana; Seth, Sahil; Spencer, Nakia D; Suzuki, Erika; Williams, Christopher C; Yu, Simon S; Zuniga, Andy M; Draetta, Giulio F; Marszalek, Joseph R; Heffernan, Timothy P; Kohl, Nancy E; Jones, Philip

NOTUM inhibition increases endocortical bone formation and bone strength

NOTUM 抑制可增加皮质内骨形成和骨强度

Robert Brommage, Jeff Liu, Peter Vogel, Faika Mseeh, Andrea Y Thompson, David G Potter, Melanie K Shadoan, Gwenn M Hansen, Sabrina Jeter-Jones, Jie Cui, Dawn Bright, Jennifer P Bardenhagen, Deon D Doree, Sofia Movérare-Skrtic, Karin H Nilsson, Petra Henning, Ulf H Lerner, Claes Ohlsson, Arthur T San

LP-925219 maximizes urinary glucose excretion in mice by inhibiting both renal SGLT1 and SGLT2

LP-925219 通过抑制肾脏 SGLT1 和 SGLT2 来最大程度地提高小鼠尿糖排泄量

David R Powell, Melinda G Smith, Deon D Doree, Angela L Harris, Wendy W Xiong, Faika Mseeh, Alan Wilson, Suma Gopinathan, Damaris Diaz, Nicole C Goodwin, Bryce Harrison, Eric Strobel, David B Rawlins, Ken Carson, Brian Zambrowicz, Zhi-Ming Ding

Lrp5 functions in bone to regulate bone mass

Lrp5在骨骼中发挥作用,调节骨量。

Cui, Yajun; Niziolek, Paul J; MacDonald, Bryan T; Zylstra, Cassandra R; Alenina, Natalia; Robinson, Daniel R; Zhong, Zhendong; Matthes, Susann; Jacobsen, Christina M; Conlon, Ronald A; Brommage, Robert; Liu, Qingyun; Mseeh, Faika; Powell, David R; Yang, Qi M; Zambrowicz, Brian; Gerrits, Han; Gossen, Jan A; He, Xi; Bader, Michael; Williams, Bart O; Warman, Matthew L; Robling, Alexander G

From genetic footprinting to antimicrobial drug targets: examples in cofactor biosynthetic pathways

从基因足迹分析到抗菌药物靶点:辅因子生物合成途径的实例

Gerdes, Svetlana Y; Scholle, Michael D; D'Souza, Mark; Bernal, Axel; Baev, Mark V; Farrell, Michael; Kurnasov, Oleg V; Daugherty, Matthew D; Mseeh, Faika; Polanuyer, Boris M; Campbell, John W; Anantha, Shubha; Shatalin, Konstantin Y; Chowdhury, Shamim A K; Fonstein, Michael Y; Osterman, Andrei L