Novel Analogues of (R)-5-(Methylamino)-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one (Sumanirole) Provide Clues to Dopamine D2/D3 Receptor Agonist Selectivity
(R)-5-(甲氨基)-5,6-二氢-4H-咪唑并[4,5,1-ij]喹啉-2(1H)-酮(Sumanirole)的新型类似物为多巴胺 D2/D3 受体激动剂的选择性提供线索
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5b01612
Mu-Fa Zou, Thomas M Keck, Vivek Kumar, Prashant Donthamsetti, Mayako Michino, Caitlin Burzynski, Catherine Schweppe, Alessandro Bonifazi, R Benjamin Free, David R Sibley, Aaron Janowsky, Lei Shi, Jonathan A Javitch, Amy Hauck Newman