日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

High-throughput screening identifies the activity of histone deacetylase inhibitors in patient-derived models of soft tissue sarcoma

高通量筛选鉴定组蛋白去乙酰化酶抑制剂在软组织肉瘤患者模型中的活性

Danks, Molly R; Manasterski, Piotr J; Beetham, Henry; Dawson, John C; Elliott, Richard J R; Culley, Jayne; Krishna, Rashi; Muir, Morwenna; Thomson, John P; Oswald, Ailsa J; Ewing, Ailith; Kerrison, William G J; Huang, Paul H; Nixon, Ioanna; Carragher, Neil O; Brunton, Valerie G

Genomics-led approach to drug testing in models of undifferentiated pleomorphic sarcoma

基因组学主导的药物测试方法在未分化多形性肉瘤模型中的应用

Manasterski, Piotr J; Danks, Molly R; Thomson, John P; Muir, Morwenna; Lee, Martin; Dawson, John C; Amaral, Ana T; Diaz-Martin, Juan; Moura, David S; Martin-Broto, Javier; Alsaadi, Ali; Salter, Donald M; Oswald, Ailsa J; Grimes, Graeme; Hayward, Larry; Hupp, Ted R; Sisley, Karen; Huang, Paul H; Carragher, Neil O; Brunton, Valerie G

Rapid Discovery and Structure-Activity Relationships of Pyrazolopyrimidines That Potently Suppress Breast Cancer Cell Growth via SRC Kinase Inhibition with Exceptional Selectivity over ABL Kinase

快速发现并阐明吡唑并嘧啶类化合物的构效关系,该类化合物通过抑制SRC激酶有效抑制乳腺癌细胞生长,且对ABL激酶具有极高的选择性。

Fraser, Craig; Dawson, John C; Dowling, Reece; Houston, Douglas R; Weiss, Jason T; Munro, Alison F; Muir, Morwenna; Harrington, Lea; Webster, Scott P; Frame, Margaret C; Brunton, Valerie G; Patton, E Elizabeth; Carragher, Neil O; Unciti-Broceta, Asier

Nuclear FAK controls chemokine transcription, Tregs, and evasion of anti-tumor immunity

核FAK调控趋化因子转录、调节性T细胞(Tregs)以及肿瘤细胞逃避免疫反应。

Serrels, Alan; Lund, Tom; Serrels, Bryan; Byron, Adam; McPherson, Rhoanne C; von Kriegsheim, Alexander; Gómez-Cuadrado, Laura; Canel, Marta; Muir, Morwenna; Ring, Jennifer E; Maniati, Eleni; Sims, Andrew H; Pachter, Jonathan A; Brunton, Valerie G; Gilbert, Nick; Anderton, Stephen M; Nibbs, Robert J B; Frame, Margaret C

Transcript and protein profiling identifies signaling, growth arrest, apoptosis, and NF-κB survival signatures following GNRH receptor activation.

转录组和蛋白质组分析揭示了 GNRH 受体激活后的信号传导、生长停滞、细胞凋亡和 NF-κB 存活特征

Meyer Colette, Sims Andrew H, Morgan Kevin, Harrison Beth, Muir Morwenna, Bai Jianing, Faratian Dana, Millar Robert P, Langdon Simon P