日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Novel Corrector for Variants of SLC6A8: A Therapeutic Opportunity for Creatine Transporter Deficiency

SLC6A8 变异的新型校正剂:肌酸转运蛋白缺乏症的治疗机会

Lara N Gechijian, Giovanni Muncipinto, T Justin Rettenmaier, Matthew T Labenski, Victor Rusu, Lea Rosskamp, Leslie Conway, Daniel van Kalken, Liam Gross, Gianna Iantosca, William Crotty, Robert Mathis, Hyejin Park, Benjamin Rabin, Christina Westgate, Matthew Lyons, Chloe Deshusses, Nicholas Brandon,

Editorial: Coumarins: New synthetic approaches and new pharmacological applications

社论:香豆素:新的合成方法和新的药理学应用

Stefanachi, Angela; Muncipinto, Giovanni; Leonetti, Francesco

A twenty-year journey exploring coumarin-based derivatives as bioactive molecules

二十年来,我们一直在探索香豆素衍生物作为生物活性分子的研究历程

Pisani, Leonardo; Catto, Marco; Muncipinto, Giovanni; Nicolotti, Orazio; Carrieri, Antonio; Rullo, Mariagrazia; Stefanachi, Angela; Leonetti, Francesco; Altomare, Cosimo

Labeling Preferences of Diazirines with Protein Biomolecules

二氮杂环丙烯与蛋白质生物分子的标记偏好

West, Alexander V; Muncipinto, Giovanni; Wu, Hung-Yi; Huang, Andrew C; Labenski, Matthew T; Jones, Lyn H; Woo, Christina M

Modulators of hepatic lipoprotein metabolism identified in a search for small-molecule inducers of tribbles pseudokinase 1 expression

在寻找三联假激酶 1 表达的小分子诱导剂时发现肝脏脂蛋白代谢的调节剂

Marek M Nagiec, Adam P Skepner, Joseph Negri, Michelle Eichhorn, Nicolas Kuperwasser, Eamon Comer, Giovanni Muncipinto, Aravind Subramanian, Clary Clish, Kiran Musunuru, Jeremy R Duvall, Michael Foley, Jose R Perez, Michelle A J Palmer

Diversity-oriented synthesis-facilitated medicinal chemistry: toward the development of novel antimalarial agents

以多样性为导向的合成促进药物化学:迈向新型抗疟药物的开发

Comer, Eamon; Beaudoin, Jennifer A; Kato, Nobutaka; Fitzgerald, Mark E; Heidebrecht, Richard W; Lee, Maurice duPont 4th; Masi, Daniela; Mercier, Marion; Mulrooney, Carol; Muncipinto, Giovanni; Rowley, Ann; Crespo-Llado, Keila; Serrano, Adelfa E; Lukens, Amanda K; Wiegand, Roger C; Wirth, Dyann F; Palmer, Michelle A; Foley, Michael A; Munoz, Benito; Scherer, Christina A; Duvall, Jeremy R; Schreiber, Stuart L

Diversity-oriented synthesis yields a new drug lead for treatment of chagas disease

多样性导向合成法获得了一种治疗恰加斯病的新药先导化合物

Dandapani, Sivaraman; Germain, Andrew R; Jewett, Ivan; le Quement, Sebastian; Marie, Jean-Charles; Muncipinto, Giovanni; Duvall, Jeremy R; Carmody, Leigh C; Perez, Jose R; Engel, Juan C; Gut, Jiri; Kellar, Danielle; Siqueira-Neto, Jair Lage; McKerrow, James H; Kaiser, Marcel; Rodriguez, Ana; Palmer, Michelle A; Foley, Michael; Schreiber, Stuart L; Munoz, Benito

Synthesis and profiling of a diverse collection of azetidine-based scaffolds for the development of CNS-focused lead-like libraries

合成和分析多种基于氮杂环丁烷的骨架化合物,用于开发针对中枢神经系统的先导化合物库

Lowe, Jason T; Lee, Maurice D 4th; Akella, Lakshmi B; Davoine, Emeline; Donckele, Etienne J; Durak, Landon; Duvall, Jeremy R; Gerard, Baudouin; Holson, Edward B; Joliton, Adrien; Kesavan, Sarathy; Lemercier, Berenice C; Liu, Haibo; Marié, Jean-Charles; Mulrooney, Carol A; Muncipinto, Giovanni; Welzel-O'Shea, Morgan; Panko, Laura M; Rowley, Ann; Suh, Byung-Chul; Thomas, Meryl; Wagner, Florence F; Wei, Jingqiang; Foley, Michael A; Marcaurelle, Lisa A

Catalytic diastereoselective petasis reactions

催化非对映选择性petasis反应

Muncipinto, Giovanni; Moquist, Philip N; Schreiber, Stuart L; Schaus, Scott E

Expanding stereochemical and skeletal diversity using petasis reactions and 1,3-dipolar cycloadditions

利用petasis反应和1,3-偶极环加成反应扩展立体化学和骨架多样性

Muncipinto, Giovanni; Kaya, Taner; Wilson, J Anthony; Kumagai, Naoya; Clemons, Paul A; Schreiber, Stuart L