日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cyclic lipopeptides as membrane fusion inhibitors against SARS-CoV-2: New tricks for old dogs

环状脂肽作为抗SARS-CoV-2的膜融合抑制剂:老狗的新招式

Shekunov, Egor V; Zlodeeva, Polina D; Efimova, Svetlana S; Muryleva, Anna A; Zarubaev, Vladimir V; Slita, Alexander V; Ostroumova, Olga S

Synthesis of isomeric 4-(N-methyltetrazolylamino)-2-phenyl-4H-thiopyrano[2,3-b]quinoline-3-carbaldehydes and 4-hydroxy-2-phenyl-4H-thiopyrano[2,3-b]quinoline-3-carbaldehyde based on tandem thiol-Michael and (aza)-Morita-Baylis-Hillman reactions and an in vitro study of the activity of the obtained compounds against influenza virus

基于串联硫醇-迈克尔加成反应和(氮杂)-Morita-Baylis-Hillman反应,合成了异构体4-(N-甲基四唑氨基)-2-苯基-4H-硫代吡喃并[2,3-b]喹啉-3-甲醛和4-羟基-2-苯基-4H-硫代吡喃并[2,3-b]喹啉-3-甲醛,并体外研究了所得化合物对流感病毒的活性。

Khramchikhin, Andrey V; Skryl'nikova, Mariya А; Pavlyukova, Yuliya N; Zarubaev, Vladimir V; Esaulkova, Yana L; Muryleva, Anna А; Shmanyova, Nadezhda T; Danagulyan, Gevorg G; Ostrovskii, Vladimir А

Synthesis, structure, and antiviral properties of novel 2-adamantyl-5-aryl-2H-tetrazoles

新型2-金刚烷基-5-芳基-2H-四唑的合成、结构及抗病毒性能

Mikolaichuk, Olga V; Zarubaev, Vladimir V; Muryleva, Anna А; Esaulkova, Yana L; Spasibenko, Daria V; Batyrenko, Alina А; Kornyakov, Ilya V; Trifonov, Rostislav Е

Single-stage synthesis of heterocyclic alkaloid-like compounds from (+)-camphoric acid and their antiviral activity

由(+)-樟脑酸一步合成杂环生物碱类化合物及其抗病毒活性

Chernyshov, Vladimir V; Yarovaya, Olga I; Fadeev, Dmitry S; Gatilov, Yuriy V; Esaulkova, Yana L; Muryleva, Anna S; Sinegubova, Katherina O; Zarubaev, Vladimir V; Salakhutdinov, Nariman F