日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Guided Development of NRAS G12D Inhibitors Based on a 5‑Azaindole Core

基于5-氮杂吲哚核心的结构导向NRAS G12D抑制剂开发

Cox, Joshua B; Nair, Vinay; Mandal, Pijus; Reyna, Naphtali; Tran, Tuyen; Mustachio, Lisa Maria; Bardenhagen, Jennifer; Fawver, Janelle; Shepard, Hannah; Hickey, Anna M; Wu, Qi; Rodriguez, Christian; Yu, Fei; Phan, Phuc; Mendiola, Andrea J; Johnson, Rebecca; Thapar, Roopa; Johnson, Troy; Jiang, Yongying; Cross, Jason B; Do, Mary K Geck; Jones, Philip; Marsalek, Joseph; Heffernan, Timothy; Soth, Michael J; Nagy, Edith

Loss of ubiquitin-specific peptidase 18 destabilizes 14-3-3ζ protein and represses lung cancer metastasis

泛素特异性肽酶 18 的缺失导致 14-3-3ζ 蛋白不稳定并抑制肺癌转移

Zibo Chen, Lin Zheng, Yulong Chen, Xiuxia Liu, Masanori Kawakami, Lisa Maria Mustachio, Jason Roszik, Katherine V Ferry-Galow, Ralph E Parchment, Xin Liu, Thorkell Andresson, Gerard Duncan, Jonathan M Kurie, Jaime Rodriguez-Canales, Xi Liu, Ethan Dmitrovsky

Single-Cell Sequencing: Current Applications in Precision Onco-Genomics and Cancer Therapeutics

单细胞测序:在精准肿瘤基因组学和癌症治疗中的最新应用

Mustachio, Lisa Maria; Roszik, Jason

A Novel CDK2/9 Inhibitor CYC065 Causes Anaphase Catastrophe and Represses Proliferation, Tumorigenesis, and Metastasis in Aneuploid Cancers

新型 CDK2/9 抑制剂 CYC065 导致后期灾难并抑制非整倍体癌症的增殖、肿瘤发生和转移

Masanori Kawakami, Lisa Maria Mustachio, Yulong Chen, Zibo Chen, Xiuxia Liu, Cheng-Hsin Wei, Jason Roszik, Adam S Kittai, Alexey V Danilov, Xiaoshan Zhang, Bingliang Fang, Jing Wang, John V Heymach, Liliya Tyutyunyk-Massey, Sarah J Freemantle, Jonathan M Kurie, Xi Liu, Ethan Dmitrovsky

Targeting KRAS in Cancer: Promising Therapeutic Strategies

靶向KRAS治疗癌症:前景广阔的治疗策略

Mustachio, Lisa Maria; Chelariu-Raicu, Anca; Szekvolgyi, Lorant; Roszik, Jason

Landscape of Immune-Related Markers and Potential Therapeutic Targets in Soft Tissue Sarcoma

软组织肉瘤中免疫相关标志物及潜在治疗靶点的概况

Roszik, Jason; Mustachio, Lisa Maria; Livingston, John A; Groisberg, Roman; Carmagnani Pestana, Roberto; Subbiah, Vivek; Conley, Anthony P

The Ubiquitin-Specific Peptidase USP18 Promotes Lipolysis, Fatty Acid Oxidation, and Lung Cancer Growth

泛素特异性肽酶USP18促进脂肪分解、脂肪酸氧化和肺癌生长

Xi Liu ,Yun Lu ,Zibo Chen ,Xiuxia Liu ,Weiguo Hu ,Lin Zheng ,Yulong Chen ,Jonathan M Kurie ,Mi Shi ,Lisa Maria Mustachio ,Thorkell Adresson ,Stephen Fox ,Jason Roszik ,Masanori Kawakami ,Sarah J Freemantle ,Ethan Dmitrovsky

Usp22 Overexpression Leads to Aberrant Signal Transduction of Cancer-Related Pathways but Is Not Sufficient to Drive Tumor Formation in Mice

Usp22 过表达导致癌症相关通路信号转导异常,但不足以驱动小鼠肿瘤形成

Xianghong Kuang, Michael J McAndrew, Lisa Maria Mustachio, Ying-Jiun C Chen, Boyko S Atanassov, Kevin Lin, Yue Lu, Jianjun Shen, Andrew Salinger, Timothy Macatee, Sharon Y R Dent, Evangelia Koutelou

Targeting the SAGA and ATAC Transcriptional Coactivator Complexes in MYC-Driven Cancers

靶向 MYC 驱动的癌症中的 SAGA 和 ATAC 转录共激活复合物

Mustachio, Lisa Maria; Roszik, Jason; Farria, Aimee; Dent, Sharon Y R

Current Targeted Therapies for the Fight against Non-Small Cell Lung Cancer

目前针对非小细胞肺癌的靶向疗法

Mustachio, Lisa Maria; Roszik, Jason