Structure-Guided Development of NRAS G12D Inhibitors Based on a 5‑Azaindole Core
基于5-氮杂吲哚核心的结构导向NRAS G12D抑制剂开发
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00647
Cox, Joshua B; Nair, Vinay; Mandal, Pijus; Reyna, Naphtali; Tran, Tuyen; Mustachio, Lisa Maria; Bardenhagen, Jennifer; Fawver, Janelle; Shepard, Hannah; Hickey, Anna M; Wu, Qi; Rodriguez, Christian; Yu, Fei; Phan, Phuc; Mendiola, Andrea J; Johnson, Rebecca; Thapar, Roopa; Johnson, Troy; Jiang, Yongying; Cross, Jason B; Do, Mary K Geck; Jones, Philip; Marsalek, Joseph; Heffernan, Timothy; Soth, Michael J; Nagy, Edith