Binding to an Unusual Inactive Kinase Conformation by Highly Selective Inhibitors of Inositol-Requiring Enzyme 1α Kinase-Endoribonuclease
肌醇需要酶 1α 激酶-内切核糖核酸酶的高选择性抑制剂与异常非活性激酶构象结合
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.8b01721
Giampiero Colombano, John J Caldwell, Thomas P Matthews, Chitra Bhatia, Amar Joshi, Tatiana McHardy, Ngai Yi Mok, Yvette Newbatt, Lisa Pickard, Jade Strover, Somaieh Hedayat, Michael I Walton, Stephanie M Myers, Alan M Jones, Harry Saville, Craig McAndrew, Rosemary Burke, Suzanne A Eccles, Faith E D