日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a fluorinated macrobicyclic antibiotic through chemical synthesis

通过化学合成发现一种氟化大环双环抗生素

Tresco, Ben I C; Wu, Kelvin J Y; Ramkissoon, Antonio; Aleksandrova, Elena V; Purdy, Michael; See, Dominic N Y; Liu, Richard Y; Polikanov, Yury S; Myers, Andrew G

Why Sulfur is Important in Lincosamide Antibiotics

为什么硫在林可酰胺类抗生素中如此重要

Wu, Kelvin J Y; Aleksandrova, Elena V; Robinson, Paul J; Benedetto, Amy E; Yu, Meiyi; Tresco, Ben I C; See, Dominic N Y; Jiang, Tong; Ramkissoon, Antonio; Dunand, Clémence F; Svetlov, Maxim S; Lee, Joonho; Polikanov, Yury S; Myers, Andrew G

An antibiotic preorganized for ribosomal binding overcomes antimicrobial resistance

一种预先组织好、可与核糖体结合的抗生素能够克服抗菌素耐药性。

Wu, Kelvin J Y; Tresco, Ben I C; Ramkissoon, Antonio; Aleksandrova, Elena V; Syroegin, Egor A; See, Dominic N Y; Liow, Priscilla; Dittemore, Georgia A; Yu, Meiyi; Testolin, Giambattista; Mitcheltree, Matthew J; Liu, Richard Y; Svetlov, Maxim S; Polikanov, Yury S; Myers, Andrew G

Practical Synthesis of Macrobicyclic Thiolincosamines

大环硫代钴胺的实用合成

Wu, Kelvin J Y; Tresco, Ben I C; Xiao, Junzhe; See, Dominic N Y; Myers, Andrew G

Structural basis of Cfr-mediated antimicrobial resistance and mechanisms to evade it

Cfr介导的抗菌素耐药性的结构基础及其逃避机制

Aleksandrova, Elena V; Wu, Kelvin J Y; Tresco, Ben I C; Syroegin, Egor A; Killeavy, Erin E; Balasanyants, Samson M; Svetlov, Maxim S; Gregory, Steven T; Atkinson, Gemma C; Myers, Andrew G; Polikanov, Yury S

Synthetic lincosamides iboxamycin and cresomycin are active against ocular multidrug-resistant methicillin-resistant Staphylococcus aureus carrying erm genes

合成林可酰胺类抗生素伊博沙霉素和克瑞索霉素对携带erm基因的眼部多重耐药耐甲氧西林金黄色葡萄球菌具有活性。

André, Camille; Wu, Kelvin J Y; Myers, Andrew G; Bispo, Paulo J M

Genome-encoded ABCF factors implicated in intrinsic antibiotic resistance in Gram-positive bacteria: VmlR2, Ard1 and CplR

基因组编码的ABCF因子与革兰氏阳性菌的固有抗生素耐药性有关:VmlR2、Ard1和CplR

Obana, Nozomu; Takada, Hiraku; Crowe-McAuliffe, Caillan; Iwamoto, Mizuki; Egorov, Artyom A; Wu, Kelvin J Y; Chiba, Shinobu; Murina, Victoriia; Paternoga, Helge; Tresco, Ben I C; Nomura, Nobuhiko; Myers, Andrew G; Atkinson, Gemma C; Wilson, Daniel N; Hauryliuk, Vasili

[3+2] Dipolar Cycloaddition of a Stabilized Azomethine Ylide and an Electron-Deficient Dipolarophile: Revision of Regioselectivity

[3+2] 稳定亚胺叶立德与缺电子亲偶极体偶极环加成反应:区域选择性修正

Wu, Kelvin J Y; Benedetto, Amy E; Myers, Andrew G

A method for tritiation of iboxamycin permits measurement of its ribosomal binding

一种用于氚标记异博沙霉素的方法可以测量其核糖体结合能力。

Wu, Kelvin J Y; Klepacki, Dorota; Mankin, Alexander S; Myers, Andrew G

Structural basis of Cfr-mediated antimicrobial resistance and mechanisms for its evasion

Cfr介导的抗菌素耐药性的结构基础及其逃避机制

Aleksandrova, Elena V; Wu, Kelvin J Y; Tresco, Ben I C; Syroegin, Egor A; Killeavy, Erin E; Balasanyants, Samson M; Svetlov, Maxim S; Gregory, Steven T; Atkinson, Gemma C; Myers, Andrew G; Polikanov, Yury S