Discovery of MK-8282 as a Potent G-Protein-Coupled Receptor 119 Agonist for the Treatment of Type 2 Diabetes
发现 MK-8282 是一种强效的 G 蛋白偶联受体 119 激动剂,可用于治疗 2 型糖尿病
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.8b00073
Neelamkavil, Santhosh F; Stamford, Andrew W; Kowalski, Timothy; Biswas, Dipshikha; Boyle, Craig; Chackalamannil, Samuel; Xia, Yan; Jayne, Charles; Neustadt, Bernard; Hao, Jinsong; Liu, Hong; Dai, Xing; Baker, Hana; Hawes, Brian; O'Neill, Kim; Tang, Huadong; Greenlee, William J