日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An allosteric cyclin E-CDK2 site mapped by paralog hopping with covalent probes.

利用共价探针通过旁系同源物跃迁定位变构细胞周期蛋白 E-CDK2 位点

Zhang Yuanjin, Liu Zhonglin, Hirschi Marscha, Brodsky Oleg, Johnson Eric, Won Sang Joon, Nagata Asako, Bezwada Divya, Petroski Matthew D, Majmudar Jaimeen D, Niessen Sherry, VanArsdale Todd, Gilbert Adam M, Hayward Matthew M, Stewart Al E, Nager Andrew R, Melillo Bruno, Cravatt Benjamin F

Covalent EGFR inhibitor analysis reveals importance of reversible interactions to potency and mechanisms of drug resistance

共价EGFR抑制剂分析揭示了可逆相互作用对药物效力和耐药机制的重要性

Schwartz, Phillip A; Kuzmic, Petr; Solowiej, James; Bergqvist, Simon; Bolanos, Ben; Almaden, Chau; Nagata, Asako; Ryan, Kevin; Feng, Junli; Dalvie, Deepak; Kath, John C; Xu, Meirong; Wani, Revati; Murray, Brion William

Protein redox chemistry: post-translational cysteine modifications that regulate signal transduction and drug pharmacology

蛋白质氧化还原化学:调控信号转导和药物药理学的翻译后半胱氨酸修饰

Wani, Revati; Nagata, Asako; Murray, Brion W