日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A long-lasting PI3Kδ inhibitor zandelisib forms a water-shielded hydrogen bond with p110δ and demonstrates sustained inhibitory effects.

长效 PI3Kδ 抑制剂 zandelisib 与 p110δ 形成水屏蔽氢键,并表现出持续的抑制作用

Kunieda Kana, Nagiri Chisae, Watanabe Miwa, Yoshida Tadashi, Zou Jian, Kaneda Ayumi, Takahashi Yuichi, Aburai Kenichi, Saito Jun-Ichi, Umehara Hiroshi, Otsu Yoshiaki, Ishii Toshihiko

Structural insights into the agonist selectivity of the adenosine A(3) receptor.

腺苷 A(3) 受体激动剂选择性的结构见解

Oshima Hidetaka S, Ogawa Akiko, Sano Fumiya K, Akasaka Hiroaki, Kawakami Tomoyoshi, Iwama Aika, Okamoto Hiroyuki H, Nagiri Chisae, Wei Fan-Yan, Shihoya Wataru, Nureki Osamu

Pharmacophore-guided Virtual Screening to Identify New β(3) -adrenergic Receptor Agonists

药效团引导的虚拟筛选用于鉴定新的β(3)-肾上腺素能受体激动剂

Ujiantari, Navista Sri Octa; Ham, Seungmin; Nagiri, Chisae; Shihoya, Wataru; Nureki, Osamu; Hutchinson, Dana Sabine; Schuster, Daniela