Sulphostin-inspired N-phosphonopiperidones as selective covalent DPP8 and DPP9 inhibitors.
受磺基膦酸酯启发而合成的 N-膦酸哌啶酮类化合物作为选择性共价 DPP8 和 DPP9 抑制剂
期刊:Nature Communications
影响因子:15.7
doi:10.1038/s41467-025-58493-z
Sewald Leonard, Tabak Werner W A, Fehr Lorenz, Zolg Samuel, Najdzion Maja, Verhoef Carlo J A, Podlesainski David, Geiss-Friedlander Ruth, Lammens Alfred, Kaschani Farnusch, Hellerschmied Doris, Huber Robert, Kaiser Markus