日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inhibition of dimeric SARS-CoV-2 Mpro displays positive cooperativity and a mixture of covalent and non-covalent binding.

二聚体 SARS-CoV-2 Mpro 的抑制表现出正协同性,并且是共价和非共价结合的混合

Padmanabha Das Krishna M, Chen Jun, Charifson Paul S, Green Jeremy, Tang Henry, Panchal Sanjay, Pu Fan, Korepanova Alla, Dubey Abhinav, Afanador Gustavo, Stojkovic Vladimir, Nocek Boguslaw, Bigelow Lance, Stubbs Sarah H, Davey Robert A, DeGoey David A, Arthanari Haribabu, Namchuk Mark N

Advancing New Chemical Modalities into Clinical Studies

将新的化学疗法推进临床研究

Blanco, Maria-Jesus; Gardinier, Kevin M; Namchuk, Mark N

A review of clinical efficacy data supporting emergency use authorization for COVID-19 therapeutics and lessons for future pandemics

对支持新冠肺炎治疗药物紧急使用授权的临床疗效数据进行回顾,并从中汲取对未来大流行病的经验教训

Yoo, Seo-Hyun; Kim, Lauren; Lu, Michelle; Nagoshi, Kira; Namchuk, Mark N

A multi-pronged approach targeting SARS-CoV-2 proteins using ultra-large virtual screening

利用超大规模虚拟筛选技术,采用多管齐下的方法靶向SARS-CoV-2蛋白

Gorgulla, Christoph; Padmanabha Das, Krishna M; Leigh, Kendra E; Cespugli, Marco; Fischer, Patrick D; Wang, Zi-Fu; Tesseyre, Guilhem; Pandita, Shreya; Shnapir, Alec; Calderaio, Anthony; Gechev, Minko; Rose, Alexander; Lewis, Noam; Hutcheson, Colin; Yaffe, Erez; Luxenburg, Roni; Herce, Henry D; Durmaz, Vedat; Halazonetis, Thanos D; Fackeldey, Konstantin; Patten, J J; Chuprina, Alexander; Dziuba, Igor; Plekhova, Alla; Moroz, Yurii; Radchenko, Dmytro; Tarkhanova, Olga; Yavnyuk, Irina; Gruber, Christian; Yust, Ryan; Payne, Dave; Näär, Anders M; Namchuk, Mark N; Davey, Robert A; Wagner, Gerhard; Kinney, Jamie; Arthanari, Haribabu

A Multi-Pronged Approach Targeting SARS-CoV-2 Proteins Using Ultra-Large Virtual Screening

利用超大规模虚拟筛选技术,采用多管齐下的方法靶向SARS-CoV-2蛋白

Gorgulla, Christoph; Padmanabha Das, Krishna M; Leigh, Kendra E; Cespugli, Marco; Fischer, Patrick D; Wang, Zi-Fu; Tesseyre, Guilhem; Pandita, Shreya; Shnapir, Alec; Calderaio, Anthony; Gechev, Minko; Rose, Alexander; Lewis, Noam; Hutcheson, Colin; Yaffe, Erez; Luxenburg, Roni; Herce, Henry D; Durmaz, Vedat; Halazonetis, Thanos D; Fackeldey, Konstantin; Patten, Justin J; Chuprina, Alexander; Dziuba, Igor; Plekhova, Alla; Moroz, Yurii; Radchenko, Dmytro; Tarkhanova, Olga; Yavnyuk, Irina; Gruber, Christian; Yust, Ryan; Payne, Dave; Näär, Anders M; Namchuk, Mark N; Davey, Robert A; Wagner, Gerhard; Kinney, Jamie; Arthanari, Haribabu