日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Anti-cancer effects of 3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one derivatives on hepatocellular carcinoma harboring FGFR4 activation

3,4-二氢嘧啶并[4,5-d]嘧啶-2(1H)-酮衍生物对FGFR4活化肝细胞癌的抗癌作用

Yunju Nam, Injae Shin, Younghoon Kim, SeongShick Ryu, Namdoo Kim, Eunhye Ju, Taebo Sim

Novel NanoLuc substrates enable bright two-population bioluminescence imaging in animals

新型 NanoLuc 基质可在动物体内实现明亮的双群生物发光成像

Yichi Su #, Joel R Walker #, Yunhee Park, Thomas P Smith, Lan Xiang Liu, Mary P Hall, Louai Labanieh, Robin Hurst, David C Wang, Lance P Encell, Namdoo Kim, Feijie Zhang, Mark A Kay, Kerriann M Casey, Robbie G Majzner, Jennifer R Cochran, Crystal L Mackall, Thomas A Kirkland, Michael Z Lin5

Development of a miRNA-controlled dual-sensing system and its application for targeting miR-21 signaling in tumorigenesis

miRNA 控制的双传感系统的开发及其在肿瘤发生中靶向 miR-21 信号传导的应用

Yoona Seo, Sung Soo Kim, Namdoo Kim, Sungchan Cho, Jong Bae Park, Jong Heon Kim

An orange calcium-modulated bioluminescent indicator for non-invasive activity imaging

用于非侵入性活动成像的橙色钙调制生物发光指示器

Younghee Oh, Yunhee Park, Julia H Cho, Haodi Wu, Nicole K Paulk, Lan Xiang Liu, Namdoo Kim, Mark A Kay, Joseph C Wu, Michael Z Lin

Identification of 1 H-pyrazolo[3,4-b]pyridine derivatives as potent ALK-L1196M inhibitors

鉴定 1 H-吡唑并[3,4-b]吡啶衍生物作为有效的 ALK-L1196M 抑制剂

Yunju Nam, Dongkeun Hwang, Namdoo Kim, Hong-Seog Seo, Khalid B Selim, Taebo Sim

Development of covalent inhibitors that can overcome resistance to first-generation FGFR kinase inhibitors

开发可克服第一代 FGFR 激酶抑制剂耐药性的共价抑制剂

Li Tan, Jun Wang, Junko Tanizaki, Zhifeng Huang, Amir R Aref, Maria Rusan, Su-Jie Zhu, Yiyun Zhang, Dalia Ercan, Rachel G Liao, Marzia Capelletti, Wenjun Zhou, Wooyoung Hur, NamDoo Kim, Taebo Sim, Suzanne Gaudet, David A Barbie, Jing-Ruey Joanna Yeh, Cai-Hong Yun, Peter S Hammerman, Moosa Mohammadi,

Structural determinants for ERK5 (MAPK7) and leucine rich repeat kinase 2 activities of benzo[e]pyrimido-[5,4-b]diazepine-6(11H)-ones

苯并[e]嘧啶并[5,4-b]二氮卓-6(11H)-酮的 ERK5 (MAPK7) 和亮氨酸富集重复激酶 2 活性的结构决定因素

Xianming Deng, Jonathan M Elkins, Jinwei Zhang, Qingkai Yang, Tatiana Erazo, Nestor Gomez, Hwan Geun Choi, Jinhua Wang, Nicolas Dzamko, Jiing-Dwan Lee, Taebo Sim, NamDoo Kim, Dario R Alessi, Jose M Lizcano, Stefan Knapp, Nathanael S Gray

Discovery of potent and selective covalent inhibitors of JNK

发现强效且选择性的 JNK 共价抑制剂

Tinghu Zhang, Francisco Inesta-Vaquera, Mario Niepel, Jianming Zhang, Scott B Ficarro, Thomas Machleidt, Ting Xie, Jarrod A Marto, NamDoo Kim, Taebo Sim, John D Laughlin, Hajeung Park, Philip V LoGrasso, Matt Patricelli, Tyzoon K Nomanbhoy, Peter K Sorger, Dario R Alessi, Nathanael S Gray