日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Monovalent pseudo-natural products supercharge degradation of IDO1 by its native E3 KLHDC3.

单价伪天然产物可加速 IDO1 的天然 E3 KLHDC3 的降解。

Hennes Elisabeth, Lucas Belén, Scholes Natalie S, Cheng Xiu-Fen, Scott Daniel C, Bischoff Matthias, Reich Katharina, Gasper Raphael, Lucas María, Xu Teng Teng, Rossini Sofia, Pulvermacher Lisa-Marie, Dötsch Lara, Imrichova Hana, Brause Alexandra, Führer Siska, Naredla Kesava Reddy, Sievers Sonja, Kumar Kamal, Janning Petra, Orabona Ciriana, Gersch Malte, Murray Peter J, Schulman Brenda A, Winter Georg E, Ziegler Slava, Waldmann Herbert

Design, Synthesis, and Structural Evolution of Pseudo-Natural Product IDO1 Inhibitors and Degraders

拟天然产物IDO1抑制剂和降解剂的设计、合成和结构演变

Cheng, Xiu-Fen; Lucas, Belén; Lampe, Philipp; Ugel, Stefano; Chen, Suyuan; Unger, Anke; Bischoff, Matthias; Adariani, Soheila Rezaei; Naredla, Kesava Reddy; Kumar, Kamal; Schmidt, Annika; Strohmann, Carsten; Janning, Petra; Gasper, Raphael; Lucas, María; Gersch, Malte; Sievers, Sonja; Bronte, Vincenzo; Ziegler, Slava; Waldmann, Herbert

A Rare Case of Epithelioid Haemangioendothelioma of the Lateral Orbit in a 22-Year-Old Patient

一例罕见的发生于22岁患者的外侧眶上皮样血管内皮瘤

Abdullah, Jeffrey; Chohan, Amarpreet Kaur; Mawji, Sadiq; Naredla, Pradyumna; Idle, Matthew R

Identification of a Monovalent Pseudo-Natural Product Degrader Class Supercharging Degradation of IDO1 by its native E3 KLHDC3

鉴定出一种单价伪天然产物降解剂,该降解剂可显著增强其天然 E3 酶 KLHDC3 对 IDO1 的降解作用

Hennes, Elisabeth; Lucas, Belén; Scholes, Natalie S; Cheng, Xiu-Fen; Scott, Daniel C; Bischoff, Matthias; Reich, Katharina; Gasper, Raphael; Lucas, María; Xu, Teng Teng; Pulvermacher, Lisa-Marie; Dötsch, Lara; Imrichova, Hana; Brause, Alexandra; Naredla, Kesava Reddy; Sievers, Sonja; Kumar, Kamal; Janning, Petra; Gersch, Malte; Murray, Peter J; Schulman, Brenda A; Winter, Georg E; Ziegler, Slava; Waldmann, Herbert

Development and In Vitro Characterization of Antibiotic-Loaded Nanocarriers for Dental Delivery

用于牙科输送的载抗生素纳米载体的开发及体外表征

Mohammed Ghazwani, Rajalakshimi Vasudevan, Geetha Kandasamy, Umme Hani, Gaddam Niharika, Manusri Naredla, Praveen Devanandan, Ranadheer Chowdary Puvvada, Abdulrahman A Almehizia, Abdulrahim R Hakami, Rajeshri Dhurke

Impact of vitamin B6 deficiency on the severity of diabetic peripheral neuropathy - A cross sectional study

维生素B6缺乏对糖尿病周围神经病变严重程度的影响——一项横断面研究

Khobrani, Moteb; Kandasamy, Geetha; Vasudevan, Rajalakshimi; Alhossan, AbdulAziz; Puvvada, Ranadheer Chowdary; Devanandan, Praveen; Dhurke, Rajeshri; Naredla, Manusri

In Situ Allene Formation via Alkyne Tautomerization to Promote [4 + 2]-Cycloadditions with a Pendant Alkyne or Nitrile

通过炔烃互变异构化原位生成丙二烯,促进与侧链炔烃或腈的[4+2]环加成反应

Kraemer, Niklas; Naredla, Rajasekhar Reddy; Hoye, Thomas R

Cyclizations of phenylethyl-substituted pyridinecarboxaldehydes

苯乙基取代的吡啶甲醛的环化反应

Naredla, Rajasekhar Reddy; Klumpp, Douglas A

Preparation of sulfonamides from N-silylamines

由N-硅胺制备磺酰胺

Naredla, Rajasekhar Reddy; Klumpp, Douglas A

Preparation of Aryl-Susbstituted 2-Oxyindoles by Superelectrophilic Chemistry

利用超亲电化学方法制备芳基取代的2-氧吲哚

Naredla, Rajasekhar Reddy; Raja, Erum K; Klumpp, Douglas A