Synthesis, biological evaluation, and in silico studies of new CDK2 inhibitors based on pyrazolo[3,4-d]pyrimidine and pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine scaffold with apoptotic activity
基于吡唑并[3,4-d]嘧啶和吡唑并[4,3-e][1,2,4]三唑并[1,5-c]嘧啶骨架的新型CDK2抑制剂的合成、生物学评价和计算机模拟研究,这些抑制剂具有凋亡活性。
期刊:Journal of Enzyme Inhibition and Medicinal Chemistry
影响因子:5.4
doi:10.1080/14756366.2022.2086866
Mandour, Asmaa A; Nassar, Ibrahim F; Abdel Aal, Mohammed T; Shahin, Mahmoud A E; El-Sayed, Wael A; Hegazy, Maghawry; Yehia, Amr Mohamed; Ismail, Ahmed; Hagras, Mohamed; Elkaeed, Eslam B; Refaat, Hanan M; Ismail, Nasser S M