日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis, biological evaluation, and in silico studies of new CDK2 inhibitors based on pyrazolo[3,4-d]pyrimidine and pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine scaffold with apoptotic activity

基于吡唑并[3,4-d]嘧啶和吡唑并[4,3-e][1,2,4]三唑并[1,5-c]嘧啶骨架的新型CDK2抑制剂的合成、生物学评价和计算机模拟研究,这些抑制剂具有凋亡活性。

Mandour, Asmaa A; Nassar, Ibrahim F; Abdel Aal, Mohammed T; Shahin, Mahmoud A E; El-Sayed, Wael A; Hegazy, Maghawry; Yehia, Amr Mohamed; Ismail, Ahmed; Hagras, Mohamed; Elkaeed, Eslam B; Refaat, Hanan M; Ismail, Nasser S M

Ethyl 5-amino-1-[(4-methyl-phen-yl)sulfon-yl]-1H-pyrazole-4-carboxyl-ate.

5-氨基-1-[(4-甲基苯基)磺酰基]-1H-吡唑-4-羧酸乙酯

Elgazwy Abdel-Sattar S Hamad, Nassar Ibrahim F, Jones Peter G