Systematic Evaluation of Tyrosine Kinase Inhibitors as OATP1B1 Substrates Using a Competitive Counterflow Screen
利用竞争性逆流筛选法系统评价酪氨酸激酶抑制剂作为 OATP1B1 底物的性能
期刊:Cancer Research Communications
影响因子:3.3
doi:10.1158/2767-9764.CRC-24-0332
Drabison, Thomas; Boeckman, Mike; Yang, Yan; Huang, Kevin M; de Bruijn, Peter; Nepal, Mahesh R; Silvaroli, Josie A; Chowdhury, Anika T; Eisenmann, Eric D; Cheng, Xiaolin; Pabla, Navjotsingh; Mathijssen, Ron H J; Baker, Sharyn D; Hu, Shuiying; Sparreboom, Alex; Talebi, Zahra