日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

JHU-2545 preferentially shields salivary glands and kidneys during PSMA-targeted imaging

在PSMA靶向成像过程中,JHU-2545优先保护唾液腺和肾脏。

Nedelcovych, Michael T; Dash, Ranjeet P; Wu, Ying; Choi, Eun Yong; Lapidus, Rena S; Majer, Pavel; Jančařík, Andrej; Abou, Diane; Penet, Marie-France; Nikolopoulou, Anastasia; Amor-Coarasa, Alex; Babich, John; Thorek, Daniel L; Rais, Rana; Kratochwil, Clemens; Slusher, Barbara S

Modulation of arousal and sleep/wake architecture by M(1) PAM VU0453595 across young and aged rodents and nonhuman primates

M(1) PAM VU0453595 对幼年和老年啮齿动物以及非人灵长类动物的觉醒和睡眠/觉醒结构的调节

Gould, Robert W; Russell, Jason K; Nedelcovych, Michael T; Bubser, Michael; Blobaum, Anna L; Bridges, Thomas M; Newhouse, Paul A; Lindsley, Craig W; Conn, P Jeffrey; Nader, Michael A; Jones, Carrie K

The Novel Glutamine Antagonist Prodrug JHU395 Has Antitumor Activity in Malignant Peripheral Nerve Sheath Tumor

新型谷氨酰胺拮抗剂前药 JHU395 对恶性外周神经鞘瘤具有抗肿瘤活性

Kathryn M Lemberg, Liang Zhao, Ying Wu, Vijayabhaskar Veeravalli, Jesse Alt, Joanna Marie H Aguilar, Ranjeet P Dash, Jenny Lam, Lukáš Tenora, Chabely Rodriguez, Michael T Nedelcovych, Cory Brayton, Pavel Majer, Jaishri O Blakeley, Rana Rais, Barbara S Slusher

Looking for Drugs in All the Wrong Places: Use of GCPII Inhibitors Outside the Brain

在错误的地方寻找药物:在脑外使用 GCPII 抑制剂

James J Vornov, Diane Peters, Mike Nedelcovych, Kristen Hollinger, Rana Rais, Barbara S Slusher

JHU-083 selectively blocks glutaminase activity in brain CD11b+ cells and prevents depression-associated behaviors induced by chronic social defeat stress

JHU-083 选择性阻断脑 CD11b+ 细胞中的谷氨酰胺酶活性,并预防因慢性社交挫败压力引起的抑郁相关行为

Xiaolei Zhu, Michael T Nedelcovych, Ajit G Thomas, Yuto Hasegawa, Aisa Moreno-Megui, Wade Coomer, Varun Vohra, Atsushi Saito, Gabriel Perez, Ying Wu, Jesse Alt, Eva Prchalova, Lukáš Tenora, Pavel Majer, Rana Rais, Camilo Rojas, Barbara S Slusher, Atsushi Kamiya

Glutamine Antagonist JHU083 Normalizes Aberrant Glutamate Production and Cognitive Deficits in the EcoHIV Murine Model of HIV-Associated Neurocognitive Disorders

谷氨酰胺拮抗剂JHU083可使EcoHIV小鼠HIV相关神经认知障碍模型中异常的谷氨酸生成和认知缺陷恢复正常

Nedelcovych, Michael T; Kim, Boe-Hyun; Zhu, Xiaolei; Lovell, Lyndah E; Manning, Arena A; Kelschenbach, Jennifer; Hadas, Eran; Chao, Wei; Prchalová, Eva; Dash, Ranjeet P; Wu, Ying; Alt, Jesse; Thomas, Ajit G; Rais, Rana; Kamiya, Atsushi; Volsky, David J; Slusher, Barbara S

Pharmacokinetics of Intranasal versus Subcutaneous Insulin in the Mouse

小鼠鼻内给药与皮下给药胰岛素的药代动力学比较

Nedelcovych, Michael T; Gadiano, Alexandra J; Wu, Ying; Manning, Arena A; Thomas, Ajit G; Khuder, Saja S; Yoo, Seung-Wan; Xu, Jiadi; McArthur, Justin C; Haughey, Norman J; Volsky, David J; Rais, Rana; Slusher, Barbara S

N-(Pivaloyloxy)alkoxy-carbonyl Prodrugs of the Glutamine Antagonist 6-Diazo-5-oxo-l-norleucine (DON) as a Potential Treatment for HIV Associated Neurocognitive Disorders

谷氨酰胺拮抗剂 6-重氮-5-氧代-l-正亮氨酸 (DON) 的 N-(新戊酰氧基)烷氧基羰基前药可作为 HIV 相关神经认知障碍的潜在治疗方法

Michael T Nedelcovych, Lukáš Tenora, Boe-Hyun Kim, Jennifer Kelschenbach, Wei Chao, Eran Hadas, Andrej Jančařík, Eva Prchalová, Sarah C Zimmermann, Ranjeet P Dash, Alexandra J Gadiano, Caroline Garrett, Georg Furtmüller, Byoungchol Oh, Gerald Brandacher, Jesse Alt, Pavel Majer, David J Volsky, Rana

Enhanced Brain Delivery of 2-(Phosphonomethyl)pentanedioic Acid Following Intranasal Administration of Its γ-Substituted Ester Prodrugs

鼻内给药γ-取代酯前药后,2-(膦酰甲基)戊二酸的脑部递送增强

Nedelcovych, Michael; Dash, Ranjeet P; Tenora, Lukáš; Zimmermann, Sarah C; Gadiano, Alexandra J; Garrett, Caroline; Alt, Jesse; Hollinger, Kristen R; Pommier, Elie; Jančařík, Andrej; Rojas, Camilo; Thomas, Ajit G; Wu, Ying; Wozniak, Krystyna; Majer, Pavel; Slusher, Barbara S; Rais, Rana

State-dependent alterations in sleep/wake architecture elicited by the M4 PAM VU0467154 - Relation to antipsychotic-like drug effects

M4 PAM VU0467154 引起的睡眠/觉醒结构的状态依赖性改变 - 与抗精神病药物样作用的关系

Robert W Gould, Michael T Nedelcovych, Xuewen Gong, Erica Tsai, Michael Bubser, Thomas M Bridges, Michael R Wood, Mark E Duggan, Nicholas J Brandon, John Dunlop, Michael W Wood, Magnus Ivarsson, Meredith J Noetzel, J Scott Daniels, Colleen M Niswender, Craig W Lindsley, P Jeffrey Conn, Carrie K Jone