日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

High-throughput 3D phenotypic screening identifies repurposed MEK inhibitors as drivers of chondrogenesis for cartilage regeneration

高通量3D表型筛选鉴定出重新利用的MEK抑制剂可作为软骨形成和软骨再生的驱动因子

Hajiali, Hadi; Cholewa-Waclaw, Justyna; Ballard, Jacob; Okur, Kerime Ebrar; Elliott, Richard; Carragher, Neil O; El Haj, Alicia J

Targeting the PREX2/RAC1/PI3Kβ Signaling Axis Confers Sensitivity to Clinically Relevant Therapeutic Approaches in Melanoma

针对 PREX2/RAC1/PI3Kβ 信号轴可提高黑色素瘤临床相关治疗方法的敏感性

Catriona A Ford, Dana Koludrovic, Patricia P Centeno, Mona Foth, Elpida Tsonou, Nikola Vlahov, Nathalie Sphyris, Kathryn Gilroy, Courtney Bull, Colin Nixon, Bryan Serrels, Alison F Munro, John C Dawson, Neil O Carragher, Valeria Pavet, David C Hornigold, Philip D Dunne, Julian Downward, Heidi C E We

Drug Combinations Targeting FAK and MEK Overcomes Tumor Heterogeneity in Glioblastoma.

靶向 FAK 和 MEK 的药物组合克服了胶质母细胞瘤的肿瘤异质性

Furqan Muhammad, Elliott Richard J R, Nagle Peter W K, Dawson John C, Masalmeh Roza, Garcia Virginia Alvarez, Munro Alison F, Drake Camilla, Morrison Gillian M, Pollard Steven M, Ebner Daniel, Brunton Valerie G, Frame Margaret C, Carragher Neil O

Single-cell morphological tracking of cell states to identify small-molecule modulators of liver differentiation

单细胞形态追踪细胞状态以识别肝脏分化的小分子调节剂

Rebecca E Graham, Runshi Zheng, Jesko Wagner, Asier Unciti-Broceta, David C Hay, Stuart J Forbes, Victoria L Gadd, Neil O Carragher

High-throughput screening identifies the activity of histone deacetylase inhibitors in patient-derived models of soft tissue sarcoma

高通量筛选鉴定组蛋白去乙酰化酶抑制剂在软组织肉瘤患者模型中的活性

Danks, Molly R; Manasterski, Piotr J; Beetham, Henry; Dawson, John C; Elliott, Richard J R; Culley, Jayne; Krishna, Rashi; Muir, Morwenna; Thomson, John P; Oswald, Ailsa J; Ewing, Ailith; Kerrison, William G J; Huang, Paul H; Nixon, Ioanna; Carragher, Neil O; Brunton, Valerie G

Genomics-led approach to drug testing in models of undifferentiated pleomorphic sarcoma

基因组学主导的药物测试方法在未分化多形性肉瘤模型中的应用

Manasterski, Piotr J; Danks, Molly R; Thomson, John P; Muir, Morwenna; Lee, Martin; Dawson, John C; Amaral, Ana T; Diaz-Martin, Juan; Moura, David S; Martin-Broto, Javier; Alsaadi, Ali; Salter, Donald M; Oswald, Ailsa J; Grimes, Graeme; Hayward, Larry; Hupp, Ted R; Sisley, Karen; Huang, Paul H; Carragher, Neil O; Brunton, Valerie G

Cellular Activity of CQWW Nullomer-Derived Peptides

CQWW Nullomer衍生肽的细胞活性

Shave, Steven; Isaksson, Rebecka; Pham, Nhan T; Elliott, Richard J R; Dawson, John C; Soudant, Julius; Carragher, Neil O; Auer, Manfred

FAK modulates glioblastoma stem cell energetics via regulation of glycolysis and glutamine oxidation

FAK通过调节糖酵解和谷氨酰胺氧化来调控胶质母细胞瘤干细胞的能量代谢。

Roza H A Masalmeh ,John C Dawson ,Virginia Alvarez Garcia ,Morwenna T Muir ,Roderick N Carter ,Giles E Hardingham ,Cameron Davies ,Rosina Graham ,Alex von Kriegsheim ,Jair Marques ,Chinmayi Pednekar ,Steven M Pollard ,Neil O Carragher ,Valerie G Brunton ,Margaret C Frame

High content 3D imaging by dual-view oblique plane microscopy

双视角斜平面显微镜高内涵3D成像

Sparks, Hugh; Rowe-Brown, Leo; Alexandrov, Yuriy; Gustafsson, Nils; Dvinskikh, Liuba; Curry, Nathan; Culley, Jayne; Lee, Martin; Le Marois, Alix; Ratcliffe, Colin D H; Phillips, Thomas A; Owczarek, Claudia; Arias Garcia, Mar; Llanses, Montserrat; Suckert, Theresa; Pelletier, Joffrey; Cortina, Carme; Hong, Wenzhi; Garcia, Edwin; Xu, Zhizhen; Zhang, Shengjie; Stassi, Giorgio; Batlle, Eduard; Colombelli, Julien; Parsons, Maddy; Bakal, Chris; Carragher, Neil O; Sahai, Erik; Dunsby, Chris

Pipeline to evaluate YAP-TEAD inhibitors indicates TEAD inhibition represses NF2-mutant mesothelioma

评估 YAP-TEAD 抑制剂的研发管线表明,TEAD 抑制可抑制 NF2 突变型间皮瘤

Richard Cunningham ,Siyang Jia ,Krishna Purohit ,Michaela Noskova Fairley ,Marcin K Maniak ,Yue Lin ,Ning Sze Hui ,Rebecca E Graham ,Adriano G Rossi ,Justyna Cholewa-Waclaw ,Pierre O Bagnaninchi ,Neil O Carragher ,Carsten Gram Hansen