日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Three-Layer Transformation Strategy toward Functionalized Fused Hydantoins and Diketopiperazines

一种用于功能化稠合乙内酰脲和二酮哌嗪的三层转化策略

Giannakaki, Maria-Aikaterini; Zingiridis, Marios; Froudas, Konstantinos G; Neochoritis, Constantinos G

The Multifaceted Legacy of Thalidomide: Chemistry and Biology Driving Modern Drug Design

沙利度胺的多方面影响:化学和生物学驱动现代药物设计

Nikovia, Konstantina; Kapsalis, Michael; Georgoulakis, Michael; Panousis, Athanasios; Neochoritis, Constantinos G

Crafting Molecular Tools for 15-Lipoxygenase-1 in a Single Step

一步构建 15-脂氧合酶-1 的分子工具

Louka, Anastasia; Spacho, Ntaniela; Korovesis, Dimitris; Adamis, Konstantinos; Papadopoulos, Christos; Kalaitzaki, Eirini-Eleni; Tavernarakis, Nektarios; Neochoritis, Constantinos G; Eleftheriadis, Nikolaos

Scaffold-hopping for molecular glues targeting the 14-3-3/ERα complex.

针对 14-3-3/ERα 复合物的分子胶的支架跃迁

Konstantinidou Markella, Zingiridis Marios, Pennings Marloes A M, Fragkiadakis Michael, Virta Johanna M, Revalde Jezrael L, Visser Emira J, Ottmann Christian, Brunsveld Luc, Neochoritis Constantinos G, Arkin Michelle R

Navigating Unexplored Territories of the Interrupted Ugi and Passerini Reactions toward Peptidomimetics

探索中断的 Ugi 和 Passerini 反应对肽模拟物的未知领域

Anastasiou, Paraskevi-Kleio; Fragkiadakis, Michael; Thomaidi, Maria; Froudas, Konstantinos G; Neochoritis, Constantinos G

The Evolution of Fluorescein into A Potential Theranostic Tool

荧光素向潜在诊疗工具的演变

Adamis, Konstantinos S; Georgoulakis, Michail; Angelonidis, Ioannis; Korovesis, Dimitris; Papadopoulos, Christos; Kapsalis, Michael; Tavernarakis, Nektarios; Eleftheriadis, Nikolaos; Neochoritis, Constantinos G

Heteroannulations of cyanoacetamide-based MCR scaffolds utilizing formamide

利用甲酰胺对氰基乙酰胺基MCR支架进行杂环化反应

Zingiridis, Marios; Papachristodoulou, Danae; Menegaki, Despoina; Froudas, Konstantinos G; Neochoritis, Constantinos G

Potential binding modes of the gut bacterial metabolite, 5-hydroxyindole, to the intestinal L-type calcium channels and its impact on the microbiota in rats

肠道细菌代谢物 5-羟基吲哚与肠道 L 型钙通道的潜在结合方式及其对大鼠微生物群的影响

Barbora Waclawiková, Paulo Cesar Telles de Souza, Markus Schwalbe, Constantinos G Neochoritis, Warner Hoornenborg, Sieger A Nelemans, Siewert J Marrink, Sahar El Aidy

Design, Synthesis, and Biological Evaluation of 2-Hydroxy-4-phenylthiophene-3-carbonitrile as PD-L1 Antagonist and Its Comparison to Available Small Molecular PD-L1 Inhibitors

2-羟基-4-苯基噻吩-3-腈作为 PD-L1 拮抗剂的设计、合成和生物学评价及其与现有小分子 PD-L1 抑制剂的比较

Marta A Ważyńska, Roberto Butera, Marta Requesens, Annechien Plat, Tryfon Zarganes-Tzitzikas, Constantinos G Neochoritis, Jacek Plewka, Lukasz Skalniak, Justyna Kocik-Krol, Bogdan Musielak, Katarzyna Magiera-Mularz, Ismael Rodriguez, Simon N Blok, Marco de Bruyn, Hans W Nijman, Philip H Elsinga, Tad

Supported Gold Nanoparticle-Catalyzed Selective Reduction of Multifunctional, Aromatic Nitro Precursors into Amines and Synthesis of 3,4-Dihydroquinoxalin-2-Ones

负载型金纳米粒子催化多功能芳香硝基前体选择性还原为胺类化合物及3,4-二氢喹喔啉-2-酮的合成

Iordanidou, Domna; Kallitsakis, Michael G; Tzani, Marina A; Ioannou, Dimitris I; Zarganes-Tzitzikas, Tryfon; Neochoritis, Constantinos G; Dömling, Alexander; Terzidis, Michael A; Lykakis, Ioannis N