日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Three-Layer Transformation Strategy toward Functionalized Fused Hydantoins and Diketopiperazines

一种用于功能化稠合乙内酰脲和二酮哌嗪的三层转化策略

Giannakaki, Maria-Aikaterini; Zingiridis, Marios; Froudas, Konstantinos G; Neochoritis, Constantinos G

The Multifaceted Legacy of Thalidomide: Chemistry and Biology Driving Modern Drug Design

沙利度胺的多方面影响:化学和生物学驱动现代药物设计

Nikovia, Konstantina; Kapsalis, Michael; Georgoulakis, Michael; Panousis, Athanasios; Neochoritis, Constantinos G

Crafting Molecular Tools for 15-Lipoxygenase-1 in a Single Step

一步构建 15-脂氧合酶-1 的分子工具

Louka, Anastasia; Spacho, Ntaniela; Korovesis, Dimitris; Adamis, Konstantinos; Papadopoulos, Christos; Kalaitzaki, Eirini-Eleni; Tavernarakis, Nektarios; Neochoritis, Constantinos G; Eleftheriadis, Nikolaos

Scaffold-hopping for molecular glues targeting the 14-3-3/ERα complex.

针对 14-3-3/ERα 复合物的分子胶的支架跃迁

Konstantinidou Markella, Zingiridis Marios, Pennings Marloes A M, Fragkiadakis Michael, Virta Johanna M, Revalde Jezrael L, Visser Emira J, Ottmann Christian, Brunsveld Luc, Neochoritis Constantinos G, Arkin Michelle R

Navigating Unexplored Territories of the Interrupted Ugi and Passerini Reactions toward Peptidomimetics

探索中断的 Ugi 和 Passerini 反应对肽模拟物的未知领域

Anastasiou, Paraskevi-Kleio; Fragkiadakis, Michael; Thomaidi, Maria; Froudas, Konstantinos G; Neochoritis, Constantinos G

The Evolution of Fluorescein into A Potential Theranostic Tool

荧光素向潜在诊疗工具的演变

Adamis, Konstantinos S; Georgoulakis, Michail; Angelonidis, Ioannis; Korovesis, Dimitris; Papadopoulos, Christos; Kapsalis, Michael; Tavernarakis, Nektarios; Eleftheriadis, Nikolaos; Neochoritis, Constantinos G

Heteroannulations of cyanoacetamide-based MCR scaffolds utilizing formamide

利用甲酰胺对氰基乙酰胺基MCR支架进行杂环化反应

Zingiridis, Marios; Papachristodoulou, Danae; Menegaki, Despoina; Froudas, Konstantinos G; Neochoritis, Constantinos G

Supported Gold Nanoparticle-Catalyzed Selective Reduction of Multifunctional, Aromatic Nitro Precursors into Amines and Synthesis of 3,4-Dihydroquinoxalin-2-Ones

负载型金纳米粒子催化多功能芳香硝基前体选择性还原为胺类化合物及3,4-二氢喹喔啉-2-酮的合成

Iordanidou, Domna; Kallitsakis, Michael G; Tzani, Marina A; Ioannou, Dimitris I; Zarganes-Tzitzikas, Tryfon; Neochoritis, Constantinos G; Dömling, Alexander; Terzidis, Michael A; Lykakis, Ioannis N

Multicomponent reaction-derived covalent inhibitor space

多组分反应衍生的共价抑制剂空间

Sutanto, Fandi; Shaabani, Shabnam; Neochoritis, Constantinos G; Zarganes-Tzitzikas, Tryfon; Patil, Pravin; Ghonchepour, Ehsan; Dömling, Alexander

TEAD-YAP Interaction Inhibitors and MDM2 Binders from DNA-Encoded Indole-Focused Ugi Peptidomimetics

来自DNA编码的吲哚靶向Ugi肽模拟物的TEAD-YAP相互作用抑制剂和MDM2结合剂

Kunig, Verena B K; Potowski, Marco; Akbarzadeh, Mohammad; Klika Škopić, Mateja; Dos Santos Smith, Denise; Arendt, Lukas; Dormuth, Ina; Adihou, Hélène; Andlovic, Blaž; Karatas, Hacer; Shaabani, Shabnam; Zarganes-Tzitzikas, Tryfon; Neochoritis, Constantinos G; Zhang, Ran; Groves, Matthew; Guéret, Stéphanie M; Ottmann, Christian; Rahnenführer, Jörg; Fried, Roland; Dömling, Alexander; Brunschweiger, Andreas