日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tailoring cariprazine for dual disorders via secondary pharmacophore optimization

通过二级药效团优化来定制卡利拉嗪用于治疗双重疾病

Vogt, Caleb D; Sanchez, Julie; Bonifazi, Alessandro; Saab, Elizabeth; Ranjit, Arina; Rais, Rana; Lane, J Robert; Newman, Amy Hauck

Revealing the location and dynamics of a concealed binding site in the dopamine transporter.

揭示多巴胺转运蛋白中隐藏结合位点的位置和动态

Zhu Rong, Sandtner Walter, Stockner Thomas, Heilinger Alexander, Holy Marion, Kudlacek Oliver, Wildling Linda, Saha Kusumika, Fröhlich Anna Sophie, Bindl Michael, Tziortzouda Paraskevi, Haider Anna, Gobl Julia, Suh Saanfor Hubert, Khan Jawad Akbar, Bicher Julia, Kastner Nina, Ebner Andreas, Gruber Hermann J, Freissmuth Michael, Newman Amy Hauck, Sitte Harald H, Hinterdorfer Peter

RDS-04-010: a novel atypical DAT inhibitor that inhibits cocaine taking and seeking and itself has low abuse potential in experimental animals

RDS-04-010:一种新型非典型DAT抑制剂,可抑制可卡因的摄入和渴求,且自身在实验动物中滥用潜力较低。

Soler-Cedeno, Omar; Galaj, Ewa; Klein, Benjamin; Cao, Jianjing; Bi, Guo-Hua; Newman, Amy Hauck; Xi, Zheng-Xiong

Development of a HiBiT Peptide-Based NanoBRET Ligand Binding Assay for Galanin Receptor 1 in Live Cells

开发基于HiBiT肽的NanoBRET配体结合分析方法用于活细胞中Galanin受体1的检测

Zhu, Hu; Daly, Harrison C; Yang, Tae Gyun; Born, Josh; Camacho-Hernandez, Gisela Andrea; Yuan, Mingyang; Inglese, Mari; Chenniappan, Vinoth Kumar; Zimmerman, Kris; Hurst, Robin; Hu, Xin; Newman, Amy Hauck; Ferré, Sergi; Ohana, Rachel Friedman; Hall, Matthew D; Patnaik, Samarjit

Contrasting the reinforcing effects of the novel dopamine transport inhibitors JJC8-088 and JJC8-091 in monkeys: Potential translation to medication assisted treatment

对比新型多巴胺转运抑制剂 JJC8-088 和 JJC8-091 在猴子体内的强化作用:潜在的药物辅助治疗转化应用

Allen, Mia I; Rahimi, Omeed; Johnson, Bernard N; Cao, Jianjing; Newman, Amy Hauck; Nader, Michael A

Presynaptic and Postsynaptic Mesolimbic Dopamine D(3) Receptors Play Distinct Roles in Cocaine Versus Opioid Reward in Mice

小鼠中突触前和突触后中脑边缘多巴胺D(3)受体在可卡因和阿片类药物奖赏中发挥不同的作用

Xi, Zheng-Xiong; Bocarsly, Miriam E; Galaj, Ewa; Hempel, Briana; Teresi, Catherine; Shaw, Marlisa; Bi, Guo-Hua; Jordan, Chloe; Linz, Emily; Alton, Hannah; Tanda, Gianluigi; Freyberg, Zachary; Alvarez, Veronica A; Newman, Amy Hauck

Development of a Fluorescently Labeled Ligand for Rapid Detection of DAT in Human and Mouse Peripheral Blood Monocytes

开发一种用于快速检测人和小鼠外周血单核细胞中DAT的荧光标记配体

Camacho-Hernandez, Gisela Andrea; Gopinath, Adithya; Okorom, Amarachi V; Khoshbouei, Habibeh; Newman, Amy Hauck

Development of Novel Tools for Dissection of Central Versus Peripheral Dopamine D2-Like Receptor Signaling in Dysglycemia

开发用于解析中枢与外周多巴胺D2样受体信号传导在血糖异常中作用的新工具

Bonifazi, Alessandro; Ellenberger, Michael; Farino, Zachary J; Aslanoglou, Despoina; Rais, Rana; Pereira, Sandra; Mantilla-Rivas, José O; Boateng, Comfort A; Eshleman, Amy J; Janowsky, Aaron; Hahn, Margaret K; Schwartz, Gary J; Slusher, Barbara S; Newman, Amy Hauck; Freyberg, Zachary

Modifications to 1-(4-(2-Bis(4-fluorophenyl)methyl)sulfinyl)alkyl Alicyclic Amines That Improve Metabolic Stability and Retain an Atypical DAT Inhibitor Profile

对 1-(4-(2-双(4-氟苯基)甲基)亚磺酰基)烷基脂环胺进行修饰,以提高其代谢稳定性并保持非典型 DAT 抑制剂特性

Okorom, Amarachi V; Camacho-Hernandez, Gisela Andrea; Salomon, Kristine; Lee, Kuo Hao; Ku, Therese C; Cao, Jianjing; Won, Sung Joon; Friedman, Jacob; Lam, Jenny; Paule, James; Rais, Rana; Klein, Benjamin; Xi, Zheng-Xiong; Shi, Lei; Loland, Claus J; Newman, Amy Hauck

Involvement of dopamine D3 receptor in impulsive choice decision-making in male rats

多巴胺D3受体参与雄性大鼠的冲动性选择决策

Shen, Hui; Ma, Zilu; Hans, Emma; Duan, Ying; Bi, Guo-Hua; Chae, Yurim C; Bonifazi, Alessandro; Battiti, Francisco O; Newman, Amy Hauck; Xi, Zheng-Xiong; Yang, Yihong