日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

SLC45A4 is a pain gene encoding a neuronal polyamine transporter

SLC45A4 是一种疼痛基因,编码神经元多胺转运蛋白。

Middleton, Steven J; Markússon, Sigurbjörn; Åkerlund, Mikael; Deme, Justin C; Tseng, Mandy; Li, Wenqianglong; Zuberi, Sana R; Kuteyi, Gabriel; Sarkies, Peter; Baskozos, Georgios; Perez-Sanchez, Jimena; Farah, Adham; Hébert, Harry L; Toikumo, Sylvanus; Yu, Zhanru; Maxwell, Susan; Dong, Yin Y; Kessler, Benedikt M; Kranzler, Henry R; Linley, John E; Smith, Blair H; Lea, Susan M; Parker, Joanne L; Lyssenko, Valeriya; Newstead, Simon; Bennett, David L

Cryo-EM structure of the human THIK-1 K2P K(+) channel reveals a lower Y gate regulated by lipids and anesthetics

人THIK-1 K2P K(+)通道的冷冻电镜结构揭示了一个受脂质和麻醉剂调控的较低Y门控

Rödström, Karin E J; Eymsh, Bisher; Proks, Peter; Hayre, Mehtab S; Cordeiro, Sönke; Mendez-Otalvaro, Edward; Madry, Christian; Rowland, Anna; Kopec, Wojciech; Newstead, Simon; Baukrowitz, Thomas; Schewe, Marcus; Tucker, Stephen J

Defined roles for the Staphylococcus aureus POT transporter DtpT in di/tripeptide uptake and glutathione utilisation inside human macrophages

金黄色葡萄球菌 POT 转运蛋白 DtpT 在人巨噬细胞内二肽/三肽摄取和谷胱甘肽利用中的作用已明确。

Khan, Imran; MacDonald, Sandy J; Markússon, Sigurbjörn; Kies, Paige J; Kraemer-Zimpel, Cristina; Robson, Callum; Parker, Joanne L; Newstead, Simon; Boucher, Dave; Hammer, Neal D; Van Der Woude, Marjan; Thomas, Gavin H

Structures of TASK-1 and TASK-3 K2P channels provide insight into their gating and dysfunction in disease.

TASK-1 和 TASK-3 K2P 通道的结构揭示了它们在疾病中的门控和功能障碍

Hall Peter Rory, Jouen-Tachoire Thibault, Schewe Marcus, Proks Peter, Baukrowitz Thomas, Carpenter Elisabeth P, Newstead Simon, Rödström Karin E J, Tucker Stephen J

Lysosomal Ion Channels and Transporters: Recent Findings, Therapeutic Potential, and Technical Approaches

溶酶体离子通道和转运蛋白:最新发现、治疗潜力和技术方法

Kondratskyi, Artem; Bazzone, Andre; Rapedius, Markus; Zerlotti, Rocco; Masson, Bastien; Sadanandan, Nidish Ponath; Parker, Joanne L; Santinho, Alexandre; Moutia, Marine; Thiam, Abdou Rachid; Kemp, Arlene; Seibertz, Fitzwilliam; Murciano, Nicoletta; Friis, Søren; Becker, Nadine; Obergrussberger, Alison; Barthmes, Maria; George, Cecilia; George, Michael; Dalrymple, David; Gasnier, Bruno; Newstead, Simon; Grimm, Christian; Fertig, Niels

Structural basis for transport and inhibition of nucleotide sugar transport in pathogenic fungi

致病真菌中核苷酸糖转运和抑制的结构基础

Parker, Joanne L; Deme, Justin C; Feddersen, Bjarne; Lea, Susan M; Newstead, Simon

Mechanism of phosphoinositide regulation of lysosomal pH via inhibition of CLC-7

磷脂酰肌醇通过抑制CLC-7调节溶酶体pH值的机制

Hilton, Jacob K; Lin, Yifei; Sefah, Eric; Deme, Justin C; Parker, Joanne L; Langton, Matthew J; Grabe, Michael; Lea, Susan; Newstead, Simon; Mindell, Joseph A

Extracellular modulation of TREK-2 activity with nanobodies provides insight into the mechanisms of K2P channel regulation

利用纳米抗体对TREK-2活性进行细胞外调控,有助于深入了解K2P通道调控机制。

Rödström, Karin E J; Cloake, Alexander; Sörmann, Janina; Baronina, Agnese; Smith, Kathryn H M; Pike, Ashley C W; Ang, Jackie; Proks, Peter; Schewe, Marcus; Holland-Kaye, Ingelise; Bushell, Simon R; Elliott, Jenna; Pardon, Els; Baukrowitz, Thomas; Owens, Raymond J; Newstead, Simon; Steyaert, Jan; Carpenter, Elisabeth P; Tucker, Stephen J

The mechanism of mammalian proton-coupled peptide transporters

哺乳动物质子偶联肽转运体的机制

Lichtinger, Simon M; Parker, Joanne L; Newstead, Simon; Biggin, Philip C

Identification of SLC45A4 as a pain gene encoding a neuronal polyamine transporter

鉴定出 SLC45A4 为编码神经元多胺转运蛋白的疼痛基因

Middleton, Steven J; Markússon, Sigurbjörn; Åkerlund, Mikael; Deme, Justin C; Tseng, Mandy; Li, Wenqianglong; Zuberi, Sana R; Kuteyi, Gabriel; Sarkies, Peter; Baskozos, Georgios; Perez-Sanchez, Jimena; Hébert, Harry L; Toikumo, Sylvanus; Farah, Adham; Maxwell, Susan; Dong, Yin Y; Kranzler, Henry R; Linley, John E; Smith, Blair H; Lea, Susan M; Parker, Joanne L; Lyssenko, Valeriya; Newstead, Simon; Bennett, David L