日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Radiation induces ESCRT pathway dependent CD44v3+ extracellular vesicle production stimulating pro-tumor fibroblast activity in breast cancer

放射线诱导ESCRT通路依赖性CD44v3+细胞外囊泡的产生,从而刺激乳腺癌中促肿瘤成纤维细胞的活性。

Gene Chatman Clark ,James David Hampton ,Jennifer E Koblinski ,Bridget Quinn ,Sitara Mahmoodi ,Olga Metcalf ,Chunqing Guo ,Erica Peterson ,Paul B Fisher ,Nicholas P Farrell ,Xiang-Yang Wang ,Ross B Mikkelsen

Suppression of RAF/MEK or PI3K synergizes cytotoxicity of receptor tyrosine kinase inhibitors in glioma tumor-initiating cells

RAF/MEK 或 PI3K 的抑制可协同增强受体酪氨酸激酶抑制剂在胶质瘤肿瘤起始细胞中的细胞毒性

Takashi Shingu, Lindsay Holmes, Verlene Henry, Qianghu Wang, Khatri Latha, Anupama E Gururaj, Laura A Gibson, Tiffany Doucette, Frederick F Lang, Ganesh Rao, Liang Yuan, Erik P Sulman, Nicholas P Farrell, Waldemar Priebe, Kenneth R Hess, Yaoqi A Wang, Jian Hu, Oliver Bögler3

Inhibition of nuclear factor kappaB proteins-platinated DNA interactions correlates with cytotoxic effectiveness of the platinum complexes

核因子 κB 蛋白-铂化 DNA 相互作用的抑制与铂配合物的细胞毒作用相关

Viktor Brabec, Jana Kasparkova, Hana Kostrhunova, Nicholas P Farrell

Nucleolar targeting by platinum: p53-independent apoptosis follows rRNA inhibition, cell-cycle arrest, and DNA compaction

铂类靶向核仁:rRNA 抑制、细胞周期停滞和 DNA 压缩后导致 p53 独立的细胞凋亡

Erica J Peterson, Vijay R Menon, Laura Gatti, Ralph Kipping, Dilhara Dewasinghe, Paola Perego, Lawrence F Povirk, Nicholas P Farrell

The phosphate clamp: sequence selective nucleic acid binding profiles and conformational induction of endonuclease inhibition by cationic Triplatin complexes

磷酸盐夹:序列选择性核酸结合谱和阳离子三铂复合物对核酸内切酶抑制的构象诱导

Andreea Prisecaru, Zara Molphy, Ralph G Kipping, Erica J Peterson, Yun Qu, Andrew Kellett, Nicholas P Farrell

Ligand modulation of a dinuclear platinum compound leads to mechanistic differences in cell cycle progression and arrest

双核铂化合物的配体调节导致细胞周期进程和停滞的机制差异

Vijay R Menon, Erica J Peterson, Kristoffer Valerie, Nicholas P Farrell, Lawrence F Povirk

Heparan sulfate proteoglycan-mediated entry pathway for charged tri-platinum compounds: differential cellular accumulation mechanisms for platinum

硫酸肝素蛋白聚糖介导的带电三铂化合物进入途径:铂的差异细胞积累机制

Heveline Silva, Frédéric Frézard, Erica J Peterson, Peyman Kabolizadeh, John J Ryan, Nicholas P Farrell

Effects of noncovalent platinum drug-protein interactions on drug efficacy: use of fluorescent conjugates as probes for drug metabolism

非共价铂类药物-蛋白质相互作用对药物疗效的影响:利用荧光结合物作为药物代谢的探针

Brad T Benedetti, Erica J Peterson, Peyman Kabolizadeh, Alberto Martínez, Ralph Kipping, Nicholas P Farrell

Transferring the concept of multinuclearity to ruthenium complexes for improvement of anticancer activity

将多核性概念转移到钌配合物以提高抗癌活性

Maria G Mendoza-Ferri, Christian G Hartinger, Marco A Mendoza, Michael Groessl, Alexander E Egger, Rene E Eichinger, John B Mangrum, Nicholas P Farrell, Magdalena Maruszak, Patrick J Bednarski, Franz Klein, Michael A Jakupec, Alexey A Nazarov, Kay Severin, Bernhard K Keppler