日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A brain-penetrant P2X7R antagonist mitigates Alzheimer's disease pathology

一种能穿透血脑屏障的P2X7R拮抗剂可减轻阿尔茨海默病病理。

Turcu, Andreea L; Oken, Adam C; Griñán-Ferré, Christian; Durner, Anna; Sierra-Marquez, Juan; Hinz-Kowalik, Sonja; Nagel, Jessica; Lee, So-Deok; Tzortzini, Efpraxia; Georgiou, Kyriakos; Bhol, Mamina; Baz, Zuriñe; Llop, Jordi; Schneider, Marion; Barbaraci, Carla; Kim, Ga-Ram; Barniol-Xicota, Marta; Val, Cristina; Brea, José; Loza, M Isabel; Pérez, Belén; Naesens, Lieve; Kolocouris, Antonios; Kim, Yong-Chul; Müller, Christa E; Nicke, Annette; Pallàs, Mercè; Mansoor, Steven E; Vázquez, Santiago

A polycyclic scaffold identified by structure-based drug design effectively inhibits the human P2X7 receptor

基于结构的药物设计鉴定出的一种多环骨架能有效抑制人P2X7受体。

Oken, Adam C; Turcu, Andreea L; Tzortzini, Eva; Georgiou, Kyriakos; Nagel, Jessica; Westermann, Franka G; Barniol-Xicota, Marta; Seidler, Jonas; Kim, Ga-Ram; Lee, So-Deok; Nicke, Annette; Kim, Yong-Chul; Müller, Christa E; Kolocouris, Antonios; Vázquez, Santiago; Mansoor, Steven E

Discovery of an allosteric binding site for anthraquinones at the human P2X4 receptor

在人P2X4受体上发现蒽醌的变构结合位点

Nagel, Jessica; Namasivayam, Vigneshwaran; Weinhausen, Stephanie; Sierra-Marquez, Juan; Baqi, Younis; Al Musawi, Hashem Ali M; Abdelrahman, Aliaa; Vaaßen, Victoria J; Schlegel, Jonathan G; Taplick, Lisa; Torp, Jane; Kubicek, Jan; Maertens, Barbara; Geyer, Matthias; Claff, Tobias; Nicke, Annette; Hagelueken, Gregor; Müller, Christa E

Nanoparticle-assisted targeting of heart lesions with cardiac myofibroblasts: Combined gene and cell therapy.

利用纳米颗粒辅助靶向心肌成纤维细胞治疗心脏病变:基因和细胞联合治疗

Schiffer Miriam, Wagner Kevin, Carls Esther, Nicke Julia, Hesse Michael, Fratila Raluca M, Hildebrand Staffan, Eberbeck Dietmar, Mohr Timo, Mohammadi Mona Malek, de la Fuente Jesus Martinez, Fleischmann Bernd K, Roell Wilhelm

Call for Papers – Purinergic Signaling: Medicinal Chemistry, Biology, Pharmacology, and Translation into Diagnostic and Therapeutic Drugs

征稿启事——嘌呤能信号传导:药物化学、生物学、药理学及其在诊断和治疗药物中的转化应用

Yang, Song; Sun, Yiran; Yan, Chenchen; Müller, Christa E; Nicke, Annette; Lohr, Christian; Freichel, Marc; Guse, Andreas H

ATP-Gated P2X7-Ion Channel on Kidney-Resident Natural Killer T Cells and Memory T Cells in Intrarenal Inflammation.

肾内炎症中肾脏驻留自然杀伤T细胞和记忆T细胞上的ATP门控P2X7离子通道

Junge Marten, Liaukouskaya Nastassia, Schwarz Nicole, Pinto-Espinoza Carolina, Schaffrath Alessa Z, Rissiek Björn, Krebs Christian F, Rattay Guido, Mittrücker Hans-Willi, Tomas Nicola M, Nicke Annette, Haag Friedrich, Huber Tobias B, Meyer-Schwesinger Catherine, Koch-Nolte Friedrich, Wanner Nicola

Measurement of Oro-Cecal Transit Time in LPS-Treated Pigs Fed High and Low Fiber Diets Using the Lactose-(13)C-Ureide Test in Breath and Saliva Samples.

使用乳糖-(13)C-脲基试验测定高纤维和低纤维饮食喂养的 LPS 处理猪的口盲肠转运时间

Cavalleri Mariagrazia, Sciascia Quentin L, Görs Solvig, Vernunft Andreas, Reyer Henry, Wimmers Klaus, Zentek Jürgen, Kluess Jeannette, Dänicke Sven, Metges Cornelia C

Dietary supplementation with L-carnitine elevates intracellular carnitine levels and affects gene expression of SLC25A20 and COX4I1, as well as non-mitochondrial respiration of bovine blood cells during systemic immune challenge.

膳食补充左旋肉碱可提高细胞内肉碱水平,并影响 SLC25A20 和 COX4I1 的基因表达,以及牛血细胞在全身免疫挑战期间的非线粒体呼吸

Seemann Leonie, Kersten Susanne, Bühler Susanne, Billenkamp Fabian, Meyer Ulrich, Visscher Christian, Huber Korinna, Most Erika, Eder Klaus, Dänicke Sven, Frahm Jana

Genetic Deletion of the Purinergic Receptor P2rx7 Worsens the Phenotype of α‑Sarcoglycan Muscular Dystrophy

嘌呤能受体P2rx7基因缺失会加重α-肌聚糖型肌营养不良症的表型

Astigiano, Cecilia; Principi, Elisa; Pintus, Sara; Benzi, Andrea; Baratto, Serena; Panicucci, Chiara; Passalacqua, Mario; Sierra-Marquez, Juan; Nicke, Annette; Antonini, Francesca; Del Zotto, Genny; Cicatiello, Annunziata Gaetana; Raffaghello, Lizzia; Rezzonico Jost, Tanja; Grassi, Fabio; Bruzzone, Santina; Bruno, Claudio; Gazzerro, Elisabetta

Quincke Triad and Hepatic Artery Pseudoaneurysm Presenting to the Emergency Department: A Case Report

昆克三联征合并肝动脉假性动脉瘤急诊就诊:病例报告

Wham, Courtney; Nicke, Daria; Burman, Justin; Meller, Robert; Trivedi, Premal; Farcas, Andra