日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting RNA:protein interactions with an integrative approach leads to the identification of potent YBX1 inhibitors

采用综合方法靶向 RNA:蛋白质相互作用,鉴定出有效的 YBX1 抑制剂

Krystel El Hage, Nicolas Babault #, Olek Maciejak #, Bénédicte Desforges #, Pierrick Craveur, Emilie Steiner, Juan Carlos Rengifo-Gonzalez, Hélène Henrie, Marie-Jeanne Clement, Vandana Joshi, Ahmed Bouhss, Liya Wang, Cyril Bauvais, David Pastré

Discovery of the First-in-Class G9a/GLP Covalent Inhibitors

发现首创的 G9a/GLP 共价抑制剂

Kwang-Su Park, Yan Xiong, Hyerin Yim, Julia Velez, Nicolas Babault, Prashasti Kumar, Jing Liu, Jian Jin

Lin28, a major translation reprogramming factor, gains access to YB-1-packaged mRNA through its cold-shock domain

Lin28 是一种重要的翻译重编程因子,它通过其冷休克结构域与 YB-1 包装的 mRNA 结合。

Anastasiia Samsonova ,Krystel El Hage ,Bénédicte Desforges ,Vandana Joshi ,Marie-Jeanne Clément ,Guillaume Lambert ,Hélène Henrie ,Nicolas Babault ,Pierrick Craveur ,Rachid C Maroun ,Emilie Steiner ,Ahmed Bouhss ,Alexandre Maucuer ,Dmitry N Lyabin ,Lev P Ovchinnikov ,Loic Hamon ,David Pastré

The dynamic conformational landscape of the protein methyltransferase SETD8

蛋白质甲基转移酶SETD8的动态构象图谱

Shi Chen # ,Rafal P Wiewiora # ,Fanwang Meng ,Nicolas Babault ,Anqi Ma ,Wenyu Yu ,Kun Qian ,Hao Hu ,Hua Zou ,Junyi Wang ,Shijie Fan ,Gil Blum ,Fabio Pittella-Silva ,Kyle A Beauchamp ,Wolfram Tempel ,Hualiang Jiang ,Kaixian Chen ,Robert J Skene ,Yujun George Zheng ,Peter J Brown ,Jian Jin ,Cheng Luo ,John D Chodera ,Minkui Luo

Discovery of Bisubstrate Inhibitors of Nicotinamide N-Methyltransferase (NNMT)

发现烟酰胺N-甲基转移酶(NNMT)双底物抑制剂

Nicolas Babault, Abdellah Allali-Hassani, Fengling Li, Jie Fan, Alex Yue, Kevin Ju, Feng Liu, Masoud Vedadi, Jing Liu, Jian Jin

Multiple Cold-Water Immersions Attenuate Muscle Damage but not Alter Systemic Inflammation and Muscle Function Recovery: A Parallel Randomized Controlled Trial

多次冷水浸泡可减轻肌肉损伤,但不会改变全身炎症和肌肉功能恢复:一项平行随机对照试验

Angelina Freitas Siqueira, Amilton Vieira, Martim Bottaro, João Batista Ferreira-Júnior, Otávio de Toledo Nóbrega, Vinícius Carolino de Souza, Rita de Cássia Marqueti, Nicolas Babault, João Luiz Quagliotti Durigan

Discovery of Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase

发现 G9a 样蛋白 (GLP) 赖氨酸甲基转移酶的强效选择性抑制剂

Yan Xiong, Fengling Li, Nicolas Babault, Aiping Dong, Hong Zeng, Hong Wu, Xin Chen, Cheryl H Arrowsmith, Peter J Brown, Jing Liu, Masoud Vedadi, Jian Jin