日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

General Platform for Efficient and Modular Assembly of GalNAc-siRNA Conjugates via Primary Amines and o-Nitrobenzyl Alcohol Cyclization Photoclick Chemistry Enabling Rapid Access to Therapeutic Oligonucleotides

利用伯胺和邻硝基苄醇环化光点击化学高效模块化组装 GalNAc-siRNA 缀合物的通用平台,可快速获得治疗性寡核苷酸

Nie, Hui-Jun; Hu, Hao; Qi, Xinming; Zhou, Yin-Jue; Liu, Lu; Chen, Xiao-Hua

Chemoproteomics reveals proteome-wide covalent and non-covalent targets of withaferin A

化学蛋白质组学揭示了醉茄内酯A在蛋白质组中的共价和非共价靶点

Nie, Hui-Jun; Fu, Ying-Jie; Long, Shang; Wang, Jia-Yu; Zhao, Wen-Si; Zhai, Lin-Hui; Yang, Yin-Long; Tan, Min-Jia; Hu, Hao; Chen, Xiao-Hua

Spatiotemporal and direct capturing global substrates of lysine-modifying enzymes in living cells.

活细胞中赖氨酸修饰酶的时空直接捕获全局底物

Hu Hao, Hu Wei, Guo An-Di, Zhai Linhui, Ma Song, Nie Hui-Jun, Zhou Bin-Shan, Liu Tianxian, Jia Xinglong, Liu Xing, Yao Xuebiao, Tan Minjia, Chen Xiao-Hua

Tumor-targeted PROTAC prodrug nanoplatform enables precise protein degradation and combination cancer therapy

肿瘤靶向PROTAC前药纳米平台可实现精准的蛋白质降解和联合癌症治疗

Zou, Zhi-Feng; Yang, Lei; Nie, Hui-Jun; Gao, Jing; Lei, Shu-Min; Lai, Yi; Zhang, Fan; Wagner, Ernst; Yu, Hai-Jun; Chen, Xiao-Hua; Xu, Zhi-Ai

Light-induced primary amines and o-nitrobenzyl alcohols cyclization as a versatile photoclick reaction for modular conjugation

光诱导伯胺和邻硝基苄醇环化反应作为一种多功能的光点击反应用于模块化偶联

Guo, An-Di; Wei, Dan; Nie, Hui-Jun; Hu, Hao; Peng, Chengyuan; Li, Shao-Tong; Yan, Ke-Nian; Zhou, Bin-Shan; Feng, Lei; Fang, Chao; Tan, Minjia; Huang, Ruimin; Chen, Xiao-Hua