日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Modeling response to the KRAS-G12C inhibitor AZD4625 in KRAS(G12C) NSCLC patient-derived xenografts reveals insights into primary resistance mechanisms

在KRAS(G12C)非小细胞肺癌患者来源的异种移植模型中模拟KRAS-G12C抑制剂AZD4625的反应,揭示了原发性耐药机制的奥秘。

Rosen, Joshua C; Cao, Pinjiang; Pham, Nhu-An; Waas, Matthew; Li, Quan; Hueniken, Katrina; Wang, Mutian; Navab, Roya; Wybenga-Groot, Leanne; Radulovich, Nikolina; Niedbala, Michael; Koers, Alex; Ross, Sarah; Moran, Michael F; Sacher, Adrian; Tsao, Ming-Sound

Use of new approach methodology for hepatic safety assessment of covalent inhibitor drug candidates.

采用新的方法对共价抑制剂候选药物进行肝脏安全性评价

Amberntsson Sara, Foster Alison J, Chouhan Bhavik, Wilkinson Stephen, Harlfinger Stephanie, Smith Graham, Kettle Jason G, Niedbala Michael, Kavanagh Stefan, Williams Dominic P