日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cell membrane cholesterol affects serotonin transporter efflux due to altered transporter oligomerization

细胞膜胆固醇通过改变转运蛋白寡聚化影响血清素转运蛋白的外排。

Rudin, Deborah; Luethi, Dino; Niello, Marco; Yang, Jae-Won; Burger, Isabella; Sandtner, Walter; Birner-Gruenberger, Ruth; Schütz, Gerhard J; Sitte, Harald H

Fluorescent PyrAte-(S)-citalopram conjugates enable imaging of the serotonin transporter in living tissue

荧光标记的PyrAte-(S)-西酞普兰缀合物可用于活体组织中血清素转运蛋白的成像

Belleza, Oliver J V; Saridakis, Iakovos; Singer, Nadja K; Westergaard, Xavier; Armentia Matheu, Sergio; Lemmerer, Miran; Riomet, Margaux; Sánchez-Murcia, Pedro A; Kastner, Nina; Rukavina, Stefanie; Xiao, Yi; Jäntsch, Kathrin; Niello, Marco; Schicker, Klaus; Sulzer, David; González, Leticia; Maulide, Nuno; Sitte, Harald H

Structure-activity relationships of serotonergic 5-MeO-DMT derivatives: insights into psychoactive and thermoregulatory properties

血清素 5-MeO-DMT 衍生物的结构-活性关系:对精神活性和体温调节特性的见解

Pol Puigseslloses, Núria Nadal-Gratacós, Gabriel Ketsela, Nicola Weiss, Xavier Berzosa, Roger Estrada-Tejedor, Mohammad Nazmul Islam, Marion Holy, Marco Niello, David Pubill, Jordi Camarasa, Elena Escubedo, Harald H Sitte, Raúl López-Arnau

Identification of the potassium-binding site in serotonin transporter

血清素转运蛋白中钾结合位点的鉴定

Hellsberg, Eva; Boytsov, Danila; Chen, Qingyang; Niello, Marco; Freissmuth, Michael; Rudnick, Gary; Zhang, Yuan-Wei; Sandtner, Walter; Forrest, Lucy R

Bioisosteric analogs of MDMA: Improving the pharmacological profile?

MDMA的生物等排体类似物:能否改善其药理特性?

Alberto-Silva Ana Sofia, Hemmer Selina, Bock Hailey A, da Silva Leticia Alves, Scott Kenneth R, Kastner Nina, Bhatt Manan, Niello Marco, Jäntsch Kathrin, Kudlacek Oliver, Bossi Elena, Stockner Thomas, Meyer Markus R, McCorvy John D, Brandt Simon D, Kavanagh Pierce, Sitte Harald H

Bioisosteric analogs of MDMA with improved pharmacological profile

具有改进药理特性的MDMA生物等排体类似物

Alberto-Silva, Ana Sofia; Hemmer, Selina; Bock, Hailey A; Alves da Silva, Leticia; Scott, Kenneth R; Kastner, Nina; Bhatt, Manan; Niello, Marco; Jäntsch, Kathrin; Kudlacek, Oliver; Bossi, Elena; Stockner, Thomas; Meyer, Markus R; McCorvy, John D; Brandt, Simon D; Kavanagh, Pierce; Sitte, Harald H

Serotonin-releasing agents with reduced off-target effects

具有较低脱靶效应的血清素释放剂

Mayer, Felix P; Niello, Marco; Cintulova, Daniela; Sideromenos, Spyridon; Maier, Julian; Li, Yang; Bulling, Simon; Kudlacek, Oliver; Schicker, Klaus; Iwamoto, Hideki; Deng, Fei; Wan, Jinxia; Holy, Marion; Katamish, Rania; Sandtner, Walter; Li, Yulong; Pollak, Daniela D; Blakely, Randy D; Mihovilovic, Marko D; Baumann, Michael H; Sitte, Harald H

Persistent binding at dopamine transporters determines sustained psychostimulant effects

多巴胺转运蛋白上的持续结合决定了精神兴奋剂的持续作用

Niello, Marco; Sideromenos, Spyridon; Gradisch, Ralph; O Shea, Ronan; Schwazer, Jakob; Maier, Julian; Kastner, Nina; Sandtner, Walter; Jäntsch, Kathrin; Lupica, Carl R; Hoffman, Alexander F; Lubec, Gert; Loland, Claus J; Stockner, Thomas; Pollak, Daniela D; Baumann, Michael H; Sitte, Harald H

Development and validation of an automated microfluidic perfusion platform for parallelized screening of compounds in vitro

开发和验证用于体外化合物并行筛选的自动化微流控灌注平台

Brugnoli, Francesca R; Holy, Marion; Niello, Marco; Maier, Julian; Hanreich, Marcus; Menzel, Mario; Haberler, Matthias; Zulus, Niklas; Pickl, Thomas; Ivanova, Christa; Muiznieks, Lisa D; Garlan, Benjamin; Sitte, Harald H

The metabolic regulator USF-1 is involved in the control of affective behaviour in mice

代谢调节剂 USF-1 参与控制小鼠的情感行为

Spyros Sideromenos #, Maria Nikou #, Barbara Czuczu, Nikolas Thalheimer, Anna Gundacker, Orsolya Horvath, Laura Cuenca Rico, Peter Stöhrmann, Marco Niello, Timo Partonen, Daniela D Pollak