日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

Cell membrane cholesterol affects serotonin transporter efflux due to altered transporter oligomerization

细胞膜胆固醇通过改变转运蛋白寡聚化影响血清素转运蛋白的外排。

期刊:Molecular Psychiatry
影响因子:10.1
doi:10.1038/s41380-025-03201-y
Rudin, Deborah; Luethi, Dino; Niello, Marco; Yang, Jae-Won; Burger, Isabella; Sandtner, Walter; Birner-Gruenberger, Ruth; Schütz, Gerhard J; Sitte, Harald H
细胞生物学
代谢
发表日期：2026
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Fluorescent PyrAte-(S)-citalopram conjugates enable imaging of the serotonin transporter in living tissue

荧光标记的PyrAte-(S)-西酞普兰缀合物可用于活体组织中血清素转运蛋白的成像

期刊:Chemical Science
影响因子:7.4
doi:10.1039/d4sc06949h
Belleza, Oliver J V; Saridakis, Iakovos; Singer, Nadja K; Westergaard, Xavier; Armentia Matheu, Sergio; Lemmerer, Miran; Riomet, Margaux; Sánchez-Murcia, Pedro A; Kastner, Nina; Rukavina, Stefanie; Xiao, Yi; Jäntsch, Kathrin; Niello, Marco; Schicker, Klaus; Sulzer, David; González, Leticia; Maulide, Nuno; Sitte, Harald H
IF
发表日期：2025
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Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors

人类血清素转运蛋白的配体偶联机制能够区分底物和抑制剂。

期刊:Nature Communications
影响因子:15.7
doi:10.1038/s41467-023-44637-6
Gradisch, Ralph; Schlögl, Katharina; Lazzarin, Erika; Niello, Marco; Maier, Julian; Mayer, Felix P; Alves da Silva, Leticia; Skopec, Sophie M C; Blakely, Randy D; Sitte, Harald H; Mihovilovic, Marko D; Stockner, Thomas
发表日期：2024
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Identification of the potassium-binding site in serotonin transporter

血清素转运蛋白中钾结合位点的鉴定

期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:9.1
doi:10.1073/pnas.2319384121
Hellsberg, Eva; Boytsov, Danila; Chen, Qingyang; Niello, Marco; Freissmuth, Michael; Rudnick, Gary; Zhang, Yuan-Wei; Sandtner, Walter; Forrest, Lucy R
发表日期：2024
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Bioisosteric analogs of MDMA: Improving the pharmacological profile?

MDMA的生物等排体类似物：能否改善其药理特性？

期刊:Journal of Neurochemistry
影响因子:4
doi:10.1111/jnc.16149
Alberto-Silva Ana Sofia, Hemmer Selina, Bock Hailey A, da Silva Leticia Alves, Scott Kenneth R, Kastner Nina, Bhatt Manan, Niello Marco, Jäntsch Kathrin, Kudlacek Oliver, Bossi Elena, Stockner Thomas, Meyer Markus R, McCorvy John D, Brandt Simon D, Kavanagh Pierce, Sitte Harald H
其它
发表日期：2024
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Bioisosteric analogs of MDMA with improved pharmacological profile

具有改进药理特性的MDMA生物等排体类似物

期刊:
影响因子:
doi:10.1101/2024.04.08.588083
Alberto-Silva, Ana Sofia; Hemmer, Selina; Bock, Hailey A; Alves da Silva, Leticia; Scott, Kenneth R; Kastner, Nina; Bhatt, Manan; Niello, Marco; Jäntsch, Kathrin; Kudlacek, Oliver; Bossi, Elena; Stockner, Thomas; Meyer, Markus R; McCorvy, John D; Brandt, Simon D; Kavanagh, Pierce; Sitte, Harald H
发表日期：2024
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Serotonin-releasing agents with reduced off-target effects

具有较低脱靶效应的血清素释放剂

期刊:Molecular Psychiatry
影响因子:10.1
doi:10.1038/s41380-022-01843-w
Mayer, Felix P; Niello, Marco; Cintulova, Daniela; Sideromenos, Spyridon; Maier, Julian; Li, Yang; Bulling, Simon; Kudlacek, Oliver; Schicker, Klaus; Iwamoto, Hideki; Deng, Fei; Wan, Jinxia; Holy, Marion; Katamish, Rania; Sandtner, Walter; Li, Yulong; Pollak, Daniela D; Blakely, Randy D; Mihovilovic, Marko D; Baumann, Michael H; Sitte, Harald H
发表日期：2023
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Persistent binding at dopamine transporters determines sustained psychostimulant effects

多巴胺转运蛋白上的持续结合决定了精神兴奋剂的持续作用

期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:9.1
doi:10.1073/pnas.2114204120
Niello, Marco; Sideromenos, Spyridon; Gradisch, Ralph; O Shea, Ronan; Schwazer, Jakob; Maier, Julian; Kastner, Nina; Sandtner, Walter; Jäntsch, Kathrin; Lupica, Carl R; Hoffman, Alexander F; Lubec, Gert; Loland, Claus J; Stockner, Thomas; Pollak, Daniela D; Baumann, Michael H; Sitte, Harald H
发表日期：2023
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Development and validation of an automated microfluidic perfusion platform for parallelized screening of compounds in vitro

开发和验证用于体外化合物并行筛选的自动化微流控灌注平台

期刊:Basic & Clinical Pharmacology & Toxicology
影响因子:3.3
doi:10.1111/bcpt.13940
Brugnoli, Francesca R; Holy, Marion; Niello, Marco; Maier, Julian; Hanreich, Marcus; Menzel, Mario; Haberler, Matthias; Zulus, Niklas; Pickl, Thomas; Ivanova, Christa; Muiznieks, Lisa D; Garlan, Benjamin; Sitte, Harald H
发表日期：2023
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Occlusion of the human serotonin transporter is mediated by serotonin-induced conformational changes in the bundle domain

人类血清素转运蛋白的阻塞是由血清素诱导的束状结构域构象变化介导的。

期刊:Journal of Biological Chemistry
影响因子:3.9
doi:10.1016/j.jbc.2022.101613
Gradisch, Ralph; Szöllősi, Dániel; Niello, Marco; Lazzarin, Erika; Sitte, Harald H; Stockner, Thomas
发表日期：2022
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