日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An allosteric cyclin E-CDK2 site mapped by paralog hopping with covalent probes.

利用共价探针通过旁系同源物跃迁定位变构细胞周期蛋白 E-CDK2 位点

Zhang Yuanjin, Liu Zhonglin, Hirschi Marscha, Brodsky Oleg, Johnson Eric, Won Sang Joon, Nagata Asako, Bezwada Divya, Petroski Matthew D, Majmudar Jaimeen D, Niessen Sherry, VanArsdale Todd, Gilbert Adam M, Hayward Matthew M, Stewart Al E, Nager Andrew R, Melillo Bruno, Cravatt Benjamin F

Selective inhibitor of platelet-activating factor acetylhydrolases 1b2 and 1b3 that impairs cancer cell survival

选择性抑制血小板活化因子乙酰水解酶1b2和1b3,从而损害癌细胞存活

Chang, Jae Won; Zuhl, Andrea M; Speers, Anna E; Niessen, Sherry; Brown, Steven J; Mulvihill, Melinda M; Fan, Yi Chiao; Spicer, Timothy P; Southern, Mark; Scampavia, Louis; Fernandez-Vega, Virneliz; Dix, Melissa M; Cameron, Michael D; Hodder, Peter S; Rosen, Hugh; Nomura, Daniel K; Kwon, Ohyun; Hsu, Ku-Lung; Cravatt, Benjamin F

Preventing farnesylation of the dynein adaptor Spindly contributes to the mitotic defects caused by farnesyltransferase inhibitors

阻止动力蛋白衔接蛋白Spindly的法尼基化是法尼基转移酶抑制剂引起有丝分裂缺陷的原因之一。

Holland, Andrew J; Reis, Rita M; Niessen, Sherry; Pereira, Cláudia; Andres, Douglas A; Spielmann, H Peter; Cleveland, Don W; Desai, Arshad; Gassmann, Reto

Integrated phenotypic and activity-based profiling links Ces3 to obesity and diabetes

整合表型和活性分析表明 Ces3 与肥胖和糖尿病相关

Dominguez, Eduardo; Galmozzi, Andrea; Chang, Jae Won; Hsu, Ku-Lung; Pawlak, Joanna; Li, Weiwei; Godio, Cristina; Thomas, Jason; Partida, David; Niessen, Sherry; O'Brien, Paul E; Russell, Aaron P; Watt, Matthew J; Nomura, Daniel K; Cravatt, Benjamin F; Saez, Enrique

The intramembrane protease Sppl2a is required for B cell and DC development and survival via cleavage of the invariant chain

膜内蛋白酶Sppl2a通过切割不变链,对B细胞和树突状细胞的发育和存活至关重要。

Beisner, Daniel R; Langerak, Petra; Parker, Albert E; Dahlberg, Carol; Otero, Francella J; Sutton, Sue E; Poirot, Laurent; Barnes, Whitney; Young, Michael A; Niessen, Sherry; Wiltshire, Tim; Bodendorf, Ursula; Martoglio, Bruno; Cravatt, Benjamin; Cooke, Michael P

Direct binding of SAS-6 to ZYG-1 recruits SAS-6 to the mother centriole for cartwheel assembly

SAS-6 与 ZYG-1 的直接结合将 SAS-6 募集到母中心粒上,从而组装成车轮状结构。

Lettman, Molly M; Wong, Yao Liang; Viscardi, Valeria; Niessen, Sherry; Chen, Sheng-Hong; Shiau, Andrew K; Zhou, Huilin; Desai, Arshad; Oegema, Karen

Pseudomonas syringae pv. syringae uses proteasome inhibitor syringolin A to colonize from wound infection sites

丁香假单胞菌丁香致病变种利用蛋白酶体抑制剂丁香素A从伤口感染部位定植。

Misas-Villamil, Johana C; Kolodziejek, Izabella; Crabill, Emerson; Kaschani, Farnusch; Niessen, Sherry; Shindo, Takayuki; Kaiser, Markus; Alfano, James R; van der Hoorn, Renier A L

A chemical biology approach to interrogate quorum-sensing regulated behaviors at the molecular and cellular level

利用化学生物学方法在分子和细胞水平上研究群体感应调控行为

Lowery, Colin A; Matamouros, Susana; Niessen, Sherry; Zhu, Jie; Scolnick, Jonathan; Lively, Jenny M; Cravatt, Benjamin F; Miller, Samuel I; Kaufmann, Gunnar F; Janda, Kim D

Chemoproteomic discovery of AADACL1 as a regulator of human platelet activation

化学蛋白质组学发现AADACL1是人血小板活化的调节因子

Holly, Stephen P; Chang, Jae Won; Li, Weiwei; Niessen, Sherry; Phillips, Ryan M; Piatt, Raymond; Black, Justin L; Smith, Matthew C; Boulaftali, Yacine; Weyrich, Andrew S; Bergmeier, Wolfgang; Cravatt, Benjamin F; Parise, Leslie V

Competitive activity-based protein profiling identifies aza-β-lactams as a versatile chemotype for serine hydrolase inhibition

基于活性竞争的蛋白质谱分析表明,氮杂β-内酰胺类化合物是一种用途广泛的丝氨酸水解酶抑制剂。

Zuhl, Andrea M; Mohr, Justin T; Bachovchin, Daniel A; Niessen, Sherry; Hsu, Ku-Lung; Berlin, Jacob M; Dochnahl, Maximilian; López-Alberca, María P; Fu, Gregory C; Cravatt, Benjamin F