Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7
发现一种对组蛋白赖氨酸去甲基化酶 KDM2/7 具有高选择性的细胞活性抑制剂
期刊:Angewandte Chemie-International Edition
影响因子:16.9
doi:10.1002/anie.201706788
Gerken, Philip A; Wolstenhulme, Jamie R; Tumber, Anthony; Hatch, Stephanie B; Zhang, Yijia; Müller, Susanne; Chandler, Shane A; Mair, Barbara; Li, Fengling; Nijman, Sebastian M B; Konietzny, Rebecca; Szommer, Tamas; Yapp, Clarence; Fedorov, Oleg; Benesch, Justin L P; Vedadi, Masoud; Kessler, Benedikt M; Kawamura, Akane; Brennan, Paul E; Smith, Martin D