日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Crystal structures of agonist-bound human cannabinoid receptor CB(1)

激动剂结合的人类大麻素受体CB(1)的晶体结构

Hua, Tian; Vemuri, Kiran; Nikas, Spyros P; Wu, Yiran; Qu, Lu; Pu, Mengchen; Korde, Anisha; Jiang, Shan; Ho, Jo-Hao; Han, Gye Won; Ding, Kang; Li, Xuanxuan; Liu, Haiguang; Hanson, Michael A; Zhao, Suwen; Bohn, Laura M; Makriyannis, Alexandros; Stevens, Raymond C; Liu, Zhi-Jie

Retraction Note: Crystal structures of agonist-bound human cannabinoid receptor CB(1)

撤稿声明:激动剂结合的人类大麻素受体 CB(1) 的晶体结构

Hua, Tian; Vemuri, Kiran; Nikas, Spyros P; Laprairie, Robert B; Wu, Yiran; Qu, Lu; Pu, Mengchen; Korde, Anisha; Jiang, Shan; Ho, Jo-Hao; Han, Gye Won; Ding, Kang; Li, Xuanxuan; Liu, Haiguang; Hanson, Michael A; Zhao, Suwen; Bohn, Laura M; Makriyannis, Alexandros; Stevens, Raymond C; Liu, Zhi-Jie

Structural basis of THC analog activity at the Cannabinoid 1 receptor.

THC类似物在大麻素1受体上的活性结构基础

Thorsen Thor S, Kulkarni Yashraj, Sykes David A, Bøggild Andreas, Drace Taner, Hompluem Pattarin, Iliopoulos-Tsoutsouvas Christos, Nikas Spyros P, Daver Henrik, Makriyannis Alexandros, Nissen Poul, Gajhede Michael, Veprintsev Dmitry B, Boesen Thomas, Kastrup Jette S, Gloriam David E

Exceptionally Potent Chiral Anandamide Analogs.

超强效手性花生四烯酸乙醇胺类似物。

Georgiadis Markos-Orestis, Ferreras Elena, Ji Lipin, Ferreira Luana Assis, Hainline John, Tong Fei, Dang Vuong Q, Faragher Alexandra, Sadybekov Anastasiia V, Bohn Laura M, Katritch Vsevolod, Hohmann Andrea G, Makriyannis Alexandros, Nikas Spyros P

Novel Tetraolefinic Chain Phenyl Substituted Endocannabinoid Probes.

新型四烯烃链苯基取代内源性大麻素探针。

Georgiadis Markos-Orestis, Ji Lipin, Tong Fei, Dang Vuong Q, Ferreira Luana Assis, Faragher Alexandra, Tran Ngan, Sadybekov Anastasiia V, Ganapathy Suthakar, Zvonok Nikolai, Katritch Vsevolod, Hohmann Andrea G, Bohn Laura M, Makriyannis Alexandros, Nikas Spyros P

Chiral Me-2-arachidonoyl Glycerols: The First Potent Endocannabinoid Glyceride Templates with Stability to COX-2

手性 Me-2-花生四烯酸甘油酯:首个对 COX-2 具有稳定性的高效内源性大麻素甘油酯模板

Nikas, Spyros P; Ji, Lipin; Liu, Yingpeng; Georgiadis, Markos-Orestis; Dopeshwarkar, Amey; Straiker, Alex; Kudalkar, Shalley; Sadybekov, Anastasiia V; Dvorakova, Michaela; Katritch, Vsevolod; Mackie, Ken; Marnett, Lawrence; Makriyannis, Alexandros

Comparison of Agonist Activity between CB1 and CB2 Receptors with Orthosteric Site Mutations

CB1和CB2受体正构位点突变激动剂活性的比较

Brust, Christina A; Swanson, Matthew A; Iliopoulos Tsoutsouvas, Christos; Dimova, Snezana T; Dang, Vuong Q; Stahl, Edward L; Ho, Jo-Hao; Nikas, Spyros P; Makriyannis, Alexandros; Bohn, Laura M

Structural basis for activation of CB1 by an endocannabinoid analog

内源性大麻素类似物激活 CB1 的结构基础

Krishna Kumar, Kaavya; Robertson, Michael J; Thadhani, Elina; Wang, Haoqing; Suomivuori, Carl-Mikael; Powers, Alexander S; Ji, Lipin; Nikas, Spyros P; Dror, Ron O; Inoue, Asuka; Makriyannis, Alexandros; Skiniotis, Georgios; Kobilka, Brian

Effects of cannabinoid agonists and antagonists in male rats discriminating the synthetic cannabinoid AM2201

大麻素激动剂和拮抗剂对雄性大鼠区分合成大麻素AM2201的影响

AlKhelb, Dalal; Burke, Emily L; Zvonok, Alexander; Iliopoulos-Tsoutsouvas, Christos; Georgiadis, Markos-Orestis; Jiang, Shan; Ho, Thanh C; Nikas, Spyros P; Makriyannis, Alexandros; Desai, Rajeev I

Synthon-based ligand discovery in virtual libraries of over 11 billion compounds

基于合成子的配体发现,利用包含超过110亿种化合物的虚拟化合物库进行筛选。

Sadybekov, Arman A; Sadybekov, Anastasiia V; Liu, Yongfeng; Iliopoulos-Tsoutsouvas, Christos; Huang, Xi-Ping; Pickett, Julie; Houser, Blake; Patel, Nilkanth; Tran, Ngan K; Tong, Fei; Zvonok, Nikolai; Jain, Manish K; Savych, Olena; Radchenko, Dmytro S; Nikas, Spyros P; Petasis, Nicos A; Moroz, Yurii S; Roth, Bryan L; Makriyannis, Alexandros; Katritch, Vsevolod