日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting RET Solvent-Front Mutants with Alkynyl Nicotinamide-Based Inhibitors

利用炔基烟酰胺类抑制剂靶向RET溶剂前沿突变体

Khatri, Ujjwol; Dayal, Neetu; Hu, Xueqing; Larocque, Elizabeth; Naganna, Nimishetti; Shen, Tao; Liu, Xuan; Holtsberg, Frederick W; Aman, M Javad; Sintim, Herman O; Wu, Jie

Orally Bioavailable 4-Phenoxy-quinoline Compound as a Potent Aurora Kinase B Relocation Blocker for Cancer Treatment

口服生物利用度高的4-苯氧基喹啉化合物作为一种强效的Aurora激酶B重定位阻滞剂用于癌症治疗

Li, Jinhua; Zhang, Ting; Shi, Qiong; Lv, Gang; Zhou, Xiaohu; Choudhry, Namrta; Kalashova, Julia; Yang, Chenglu; Li, Hongmei; Long, Yan; Sakthivel, Balasubramaniyan; Nimishetti, Naganna; Liu, Hong; Allen, Thaddeus D; Zhang, Jing; Yang, Dun

Isoquinoline Antimicrobial Agent: Activity against Intracellular Bacteria and Effect on Global Bacterial Proteome

异喹啉类抗菌剂:对细胞内细菌的活性及其对细菌整体蛋白质组的影响

Karanja, Caroline W; Naganna, Nimishetti; Abutaleb, Nader S; Dayal, Neetu; Onyedibe, Kenneth I; Aryal, Uma; Seleem, Mohamed N; Sintim, Herman O

Discovery and Optimization of Seven-Membered Lactam-Based Compounds to Phenocopy the Inhibition of the Aurora Kinase B

发现和优化七元内酰胺类化合物以模拟Aurora激酶B的抑制作用

Huang, Jian; Shi, Qiong; Choudhry, Namrta; Li, Hongmei; Yang, Chenglu; Kalashova, Julia; Yan, Ziqi; Li, Jinhua; Reddy, Mallu Chenna; Gopala, Sridhar Goud; Zhang, Shenqiu; Zhang, Jing; Nimishetti, Naganna; Yang, Dun

The Phytochemical Scoulerine Inhibits Aurora Kinase Activity to Induce Mitotic and Cytokinetic Defects

植物化学物质 Scoulerine 可抑制 Aurora 激酶活性,从而诱发有丝分裂和细胞分裂缺陷

Jinhua Li, Ziqi Yan, Hongmei Li, Qiong Shi, Vidhula Ahire, Shenqiu Zhang, Naganna Nimishetti, Dun Yang, Thaddeus D Allen, Jing Zhang