日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Needle in a Radiologic Haystack: A Report of Duodenal Toothpick Perforation With Negative X-ray and CT Imaging

放射影像学中的大海捞针:一例X线和CT影像检查结果均为阴性的十二指肠牙签穿孔病例报告

Warren, Jonathan; Perera, Niresh; Lema, Flor; Shyy, William

Small molecule APOL1 inhibitors as a precision medicine approach for APOL1-mediated kidney disease

小分子APOL1抑制剂作为APOL1介导的肾脏疾病的精准治疗手段

Brandon Zimmerman # ,Leslie A Dakin # ,Anne Fortier ,Evanthia Nanou ,Angelo Blasio ,James Mann ,Howard Miller ,Marissa Fletcher ,Tiansheng Wang ,Suganthini Nanthakumar ,Gizelle McCarthy ,Caline Matar ,Prachi Matsye ,Guanyu Wang ,Phillip Snyder ,Kevin Daniel ,Harsha Swamy ,Kelly Sullivan ,Franklin Bright ,Audrey Powers ,Kevin J Gagnon ,Fan Lu ,Steven Paula ,Suvarna Khare-Pandit ,Larry Henry ,Martine Hamel ,Francois Denis ,Olivier Nicolas ,Niresh Hariparsad ,Shyamesh Kumar ,Jennifer Proctor ,Timothy Senter ,Brinley Furey ,Mark E Bunnage

Building Confidence in Physiologically Based Pharmacokinetic Modeling of CYP3A Induction Mediated by Rifampin: An Industry Perspective

建立对利福平介导的CYP3A诱导的生理药代动力学模型的信心:行业视角

Reddy, Micaela B; Cabalu, Tamara D; de Zwart, Loeckie; Ramsden, Diane; Dowty, Martin E; Taskar, Kunal S; Badée, Justine; Bolleddula, Jayaprakasam; Boulu, Laurent; Fu, Qiang; Kotsuma, Masakatsu; Leblanc, Alix F; Lewis, Gareth; Liang, Guiqing; Parrott, Neil; Pilla Reddy, Venkatesh; Prakash, Chandra; Shah, Kushal; Umehara, Kenichi; Mukherjee, Dwaipayan; Rehmel, Jessica; Hariparsad, Niresh

Advancing Predictions of Oral Drug Absorption, CYP3A4 Induction, and Transporter-Mediated Interactions Using a Human Primary Intestinal 3D Model (EpiIntestinal™)

利用人类原代肠道三维模型(EpiIntestinal™)推进口服药物吸收、CYP3A4诱导和转运体介导的相互作用的预测

Chothe, Paresh P; Whitcher-Johnstone, Andrea; Karve, Aniruddha; Ramsden, Diane; Hariparsad, Niresh

Physiologically Based Pharmacokinetic Modeling to Assess Perpetrator and Victim Cytochrome P450 2C Induction Risk

基于生理药代动力学模型评估施害者和受害者细胞色素P450 2C诱导风险

Slavsky, Marina; Karve, Aniruddha Sunil; Hariparsad, Niresh

A mismatch in enzyme-redox partnerships underlies divergent cytochrome P450 activities between human hepatocytes and microsomes

人肝细胞和微粒体中细胞色素P450活性差异的根本原因是酶-氧化还原相互作用的不匹配。

Bapiro, Tashinga E; Martin, Scott; Blacker, Thomas S; Wilkinson, Stephen D; Orton, Alexandra L; Hariparsad, Niresh; Jones, Rhys D O; Duchen, Michael R; Harlfinger, Stephanie

Synthetic chemistry enabling the discovery and development of a series of pyrazoles as HPK1 inhibitors

合成化学促进了一系列吡唑类化合物作为HPK1抑制剂的发现和开发

Metrano, Anthony J; Morrill, Lucas A; Bommakanti, Gayathri; Casella, Robert; Cook, Steve; Escobar, Randolph A; Giblin, Kathryn A; Gosselin, Eric; Grebe, Tyler; Hariparsad, Niresh; Howells, Rachel; Lamont, Gillian M; Mele, Deanna A; Pflug, Alexander; Proia, Theresa A; Rezaei, Hadi; Richter, Magdalena; Richards, Ryan; San Martin, Maryann; Schimpl, Marianne; Schuller, Alwin G; Sha, Li; Sheppeck, James E 2nd; Song, Kun; Tang, Haoran; Wagner, David J; Wang, Jianyan; Wu, Allan; Wu, Dedong; Wu, Ye; Xu, Kevin; Ye, Minwei; Shields, Jason D; Grimster, Neil P

Epidemiology and management of motorbike chain-related fingertip injuries: A retrospective study at B&B Hospital, Kathmandu

摩托车链条相关指尖损伤的流行病学及治疗:加德满都B&B医院的回顾性研究

Jaiswal, Sweta; Shrestha, Om Prasad; Regmi, Subhash; Batajoo, Santosh; Shrestha, Niresh; Banskota, Ashok Kumar

Aminobenzotriazole inhibits and induces several key drug metabolizing enzymes complicating its utility as a pan CYP inhibitor for reaction phenotyping

氨基苯并三唑可抑制和诱导几种关键的药物代谢酶,使其作为泛 CYP 抑制剂用于反应表型分析变得复杂

Krishna C Aluri, Marina Slavsky, Ying Tan, Andrea Whitcher-Johnstone, Zhoupeng Zhang, Niresh Hariparsad, Diane Ramsden

Quantitative evaluation of trastuzumab deruxtecan pharmacokinetics and pharmacodynamics in mouse models of varying degrees of HER2 expression

在不同HER2表达程度的小鼠模型中,对曲妥珠单抗德鲁替康的药代动力学和药效学进行定量评价

Vasalou, Christina; Proia, Theresa A; Kazlauskas, Laura; Przybyla, Anna; Sung, Matthew; Mamidi, Srinivas; Maratea, Kim; Griffin, Matthew; Sargeant, Rebecca; Urosevic, Jelena; Rosenbaum, Anton I; Yuan, Jiaqi; Aluri, Krishna C; Ramsden, Diane; Hariparsad, Niresh; Jones, Rhys D O; Mettetal, Jerome T