Proteomic Ligandability Maps of Spirocycle Acrylamide Stereoprobes Identify Covalent ERCC3 Degraders
螺环丙烯酰胺立体探针的蛋白质组学配体结合能力图谱鉴定共价ERCC3降解剂
期刊:Journal of the American Chemical Society
影响因子:15.6
doi:10.1021/jacs.3c13448
Liu, Zhonglin; Remsberg, Jarrett R; Li, Haoxin; Njomen, Evert; DeMeester, Kristen E; Tao, Yongfeng; Xia, Guoqin; Hayward, Rachel E; Yoo, Minjin; Nguyen, Tracey; Simon, Gabriel M; Schreiber, Stuart L; Melillo, Bruno; Cravatt, Benjamin F