日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cysteine allostery and autoinhibition govern human STING oligomer functionality.

半胱氨酸变构和自身抑制控制着人类 STING 寡聚体的功能。

Chan Rebecca, Cao Xujun, Ergun Sabrina L, Njomen Evert, Lynch Stephen R, Ritchie Christopher, Cravatt Benjamin, Li Lingyin

Tryptoline Stereoprobe Elaboration Identifies Inhibitors of the GRPEL1-HSPA9 Chaperone Complex

色氨酸立体探针的衍生化鉴定出 GRPEL1-HSPA9 分子伴侣复合物的抑制剂

Hayward, Rachel E; Berkeley, Raymond F; Gao, Zijian; Garhammer, Maximilian; Morizono, Marc A; Njomen, Evert; Li, Haoxin; DeMeester, Kristen E; Cociorva, Victor; Herzik, Mark A Jr; Hartl, F Ulrich; Melillo, Bruno; Cravatt, Benjamin F

Redirecting the pioneering function of FOXA1 with covalent small molecules.

利用共价小分子重新定向 FOXA1 的先锋功能

Won Sang Joon, Zhang Yuxiang, Reinhardt Christopher J, Hargis Lauren M, MacRae Nicole S, DeMeester Kristen E, Njomen Evert, Remsberg Jarrett R, Melillo Bruno, Cravatt Benjamin F, Erb Michael A

Proteomic Ligandability Maps of Spirocycle Acrylamide Stereoprobes Identify Covalent ERCC3 Degraders

螺环丙烯酰胺立体探针的蛋白质组学配体结合能力图谱鉴定共价ERCC3降解剂

Liu, Zhonglin; Remsberg, Jarrett R; Li, Haoxin; Njomen, Evert; DeMeester, Kristen E; Tao, Yongfeng; Xia, Guoqin; Hayward, Rachel E; Yoo, Minjin; Nguyen, Tracey; Simon, Gabriel M; Schreiber, Stuart L; Melillo, Bruno; Cravatt, Benjamin F

Chemical tools to expand the ligandable proteome: Diversity-oriented synthesis-based photoreactive stereoprobes.

扩展可配体结合蛋白质组的化学工具:基于多样性的合成的光反应立体探针

Ogasawara Daisuke, Konrad David B, Tan Zher Yin, Carey Kimberly L, Luo Jessica, Won Sang Joon, Li Haoxin, Carter Trever R, DeMeester Kristen E, Njomen Evert, Schreiber Stuart L, Xavier Ramnik J, Melillo Bruno, Cravatt Benjamin F

Chemical tools to expand the ligandable proteome: diversity-oriented synthesis-based photoreactive stereoprobes

拓展配体结合蛋白质组的化学工具:基于多样性导向合成的光反应立体探针

Ogasawara, Daisuke; Konrad, David B; Tan, Zher Yin; Carey, Kimberly L; Luo, Jessica; Won, Sang Joon; Li, Haoxin; Carter, Trever; DeMeester, Kristen E; Njomen, Evert; Schreiber, Stuart L; Xavier, Ramnik J; Melillo, Bruno; Cravatt, Benjamin F

Chemical Proteomic Discovery of Isotype-Selective Covalent Inhibitors of the RNA Methyltransferase NSUN2

利用化学蛋白质组学方法发现RNA甲基转移酶NSUN2的同工型选择性共价抑制剂

Tao, Yongfeng; Felber, Jan G; Zou, Zhongyu; Njomen, Evert; Remsberg, Jarrett R; Ogasawara, Daisuke; Ye, Chang; Melillo, Bruno; Schreiber, Stuart L; He, Chuan; Remillard, David; Cravatt, Benjamin F

Small Molecule Enhancement of 20S Proteasome Activity Targets Intrinsically Disordered Proteins

小分子增强20S蛋白酶体活性靶向固有无序蛋白

Jones, Corey L; Njomen, Evert; Sjögren, Benita; Dexheimer, Thomas S; Tepe, Jetze J