日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

First-in-Class Dual PDGFR/Carbonic Anhydrase IX/XII Inhibitors: 6,7-Dimethoxyquinoline-Sulfonamides as Promising Antileukemic Agents

首创的双重PDGFR/碳酸酐酶IX/XII抑制剂:6,7-二甲氧基喹啉磺酰胺类药物作为有前景的抗白血病药物

Roshdy, Eslam; Řezníčková, Eva; Elbadawi, Mostafa M; Celik, Ismail; Giovannuzzi, Simone; Veselá, Denisa; Vojáčková, Veronika; Krňávková, Petra; Nocentini, Alessio; Supuran, Claudiu T; Kryštof, Vladimír; Eldehna, Wagdy M; Abe, Manabu

Bacterial Carbonic Anhydrase Inhibitor CAI0019 Demonstrates Efficacy in Enterococcus faecium Septicemic Peritonitis Mouse Model While Sparing the Microbiome

细菌碳酸酐酶抑制剂 CAI0019 在粪肠球菌败血性腹膜炎小鼠模型中显示出疗效,同时不影响肠道菌群。

Abutaleb, Nader S; Holly, Katrina J; Metcalfe, Carolyn K; Abouelkhair, Ahmed A; Tharra, Prabhakara R; Shrinidhi, Annadka; Abdelsattar, Abdallah S; Burgo, Victoria; Melotte, Glory; Akin-Olabiyi, Tomi; Knoblauch, Sean; Ramaswamy, Ramanujam; Woodson, Che; Thirumalaikumar, Venkatesh P; Rodriguez, J Alejandra; Yeo, Franklin J; Snell, Olivia C; Nocentini, Alessio; Sundararajan, Anitha; Olson, Matthew R; Supuran, Claudiu T; Seleem, Mohamed N; Flaherty, Daniel P

Harnessing oligonucleotide architecture for potent multivalent inhibition of human carbonic anhydrases

利用寡核苷酸结构实现对人类碳酸酐酶的强效多价抑制

Abbass, Eslam M; Ladu, Federico; Mansot, Justine; Noël, Mathieu; Nocentini, Alessio; Sechi, Mario; Supuran, Claudiu T; Smietana, Michael; Winum, Jean-Yves

Benzoxaboroles Are Inhibitors of the η-Class Carbonic Anhydrase From Plasmodium falciparum

苯并硼氧杂环己烷是恶性疟原虫η类碳酸酐酶的抑制剂

Bonardi, Alessandro; Wein, Sharon; Mustafa, Muhamad; Cerdan, Rachel; de Luca, Viviana; Capasso, Clemente; Gratteri, Paola; Supuran, Claudiu T; Nocentini, Alessio; Winum, Jean-Yves

4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1H-indol-1-yl)benzenesulfonamide: A Novel Polypharmacology Agent to Target Carbonic Anhydrase IX and XII With Improved Selectivity, Wnt/β-Catenin Signaling Pathway, and P-Glycoprotein

4-(5-氯-3-(3,4,5-三甲氧基苯甲酰基)-1H-吲哚-1-基)苯磺酰胺:一种新型多靶点药物,可选择性地靶向碳酸酐酶IX和XII、Wnt/β-catenin信号通路以及P-糖蛋白。

Puxeddu, Michela; Bordone, Rosa; Colla, Claudia; Rotili, Gabriele; Coluccia, Antonio; Sciò, Pietro; Cuřínová, Petra; Nocentini, Alessio; Supuran, Claudiu T; Filiberti, Serena; Turati, Marta; Ronca, Roberto; Kopecka, Joanna; Riganti, Chiara; Jimenez, Lucia; Link, Wolfgang; Bigogno, Chiara; Dondio, Giulio; Barba, Martina; Canettieri, Gianluca; Silvestri, Romano; La Regina, Giuseppe

Molecular Signatures and Functional Pathways of Human Monocytes and Macrophages in Allergy: An EAACI AllergoOncology Scoping Review

人类单核细胞和巨噬细胞在过敏反应中的分子特征和功能通路:EAACI过敏肿瘤学范围综述

Bianchini, Rodolfo; Escolar-Peña, Andrea; Pick, Vanda; Poli, Aurélie; Adams, Rebecca; Basilio, José; Cari, Luigi; Chauhan, Jitesh; Chivato, Tomás; Vecillas, Leticia de Las; Delgado-Dolset, María Isabel; Escribese, Maria M; Grandits, Melanie; Bax, Heather J; Martín-Antoniano, Isabel Adoración; Martín-Cruz, Leticia; Mayerhofer, Hanna; Michelucci, Alessandro; Nocentini, Giuseppe; Osborn, Gabriel; Pablo-Torres, Carmela; Palomares, Oscar; Pascal, Mariona; Radzikowska, Urszula; Rohr-Udilova, Nataliya; Sokolowska, Milena; Bergmann, Christoph; Jensen-Jarolim, Erika; Karagiannis, Sophia N; Rebollido-Rios, Rocio; Izquierdo, Elena

Micropatterned Liquid Crystalline Networks for Multipurpose Color Pixels

用于多用途彩色像素的微图案液晶网络

Zubritskaya, Irina; Martella, Daniele; Nocentini, Sara

Imbalance of human CD4(+) T lymphocyte subsets following atrazine treatment

阿特拉津治疗后人CD4(+) T淋巴细胞亚群失衡

Alhosseini, Mahdieh Naghavi; Maddalon, Ambra; Cari, Luigi; Ronchetti, Simona; Migliorati, Graziella; Corsini, Emanuela; Nocentini, Giuseppe

Intracellular Binding of Novel Fluorinated Compounds to Carbonic Anhydrase Isoforms Explored by In-Cell (19)F NMR

利用细胞内 (19)F NMR 研究新型氟化化合物与碳酸酐酶同工酶的细胞内结合

Costantino, Azzurra; Barbieri, Letizia; Giovannuzzi, Simone; Nocentini, Alessio; Supuran, Claudiu T; Raitelaitis, Mindaugas; Nordlund, Pär; Banci, Lucia; Luchinat, Enrico

Hit-to-Lead Optimization of Acetazolamide-Based Bacterial Carbonic Anhydrase Inhibitors with Efficacy In Vivo for Treatment of Vancomycin-Resistant Enterococci Septicemia

基于乙酰唑胺的细菌碳酸酐酶抑制剂的先导化合物优化,以评估其在体内治疗耐万古霉素肠球菌败血症的疗效。

Holly, Katrina J; Tharra, Prabhakara R; Abutaleb, Nader S; Nocentini, Alessio; Abouelkhair, Ahmed A; Youse, Molly S; Marapaka, Anil Kumar; S Abdelsattar, Abdallah; An, Weiwei; Drummond, Faith L; Snell, Olivia C; Supuran, Claudiu T; Seleem, Mohamed N; Flaherty, Daniel P