Quinazolinones as Bioisosteres of Naphthoquinones: A Path to Potent HsDHODH Inhibitors with Optimized Properties
喹唑啉酮作为萘醌的生物等排体:获得具有优化性能的高效HsDHODH抑制剂的途径
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00237
Godoi, Bruna F; Bueno, Jéssica D; Silva, Wemenes J L; da Purificação, Aline D; Leite, Pedro I P; Dos Santos, Thiago; Freitas, Murillo; Silva, Daniel G; Silva, Tais C; de Moraes, Josué; Freitas, Caroline S; Mattos, Mayara; Souza, Thiago M L; Martin, Bianca A; Lopez, Renata F V; Nonato, M Cristina; Andrade, Carolina H; Emery, Flavio S