Synthesis and Pharmacological Evaluation of 6,7-Dihydro‑3H‑Oxazolo[3,4‑a]Pyrazine-5,8-Dione Compounds as Inhibitors of Phosphodiesterases 4 and 5
6,7-二氢-3H-噁唑并[3,4-a]吡嗪-5,8-二酮类化合物作为磷酸二酯酶4和5抑制剂的合成及药理学评价
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00525
Helfstein, Débora Rocha; das Virgens, Marcio Fernando; Rojas Moscoso, Julio Alejandro; Zaminelli, Tiago; Toledo, Fabiano Travanca; Maia de Lima, Jeniffer; Medeiros, Larissa Ozols; Marcello, Bianca Alves; Soares, Vinícius Marques; Passos, Gabriela Reolon; de Padua, Sarah Saraiva; Wolf, Matheus Eduardo Gonçalves; Carneiro, Leonardo Martins; De Nucci, Gilberto; Keppler, Artur Franz; Mónica, Fabíola Zakia