日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Leveraging conformational ensembles in allosteric drug discovery

利用构象集合进行变构药物发现

Nussinov, Ruth; Regev, Clil; Jang, Hyunbum

A Quantum Framework for Protein Binding-Site Structure Prediction on Utility-Level Quantum Processors

基于实用级量子处理器的蛋白质结合位点结构预测量子框架

Zhang, Yuqi; Yang, Yuxin; Martin, William; Lin, Kingsten; Wang, Zixu; Lu, Cheng-Chang; Jiang, Weiwen; Nussinov, Ruth; Loscalzo, Joseph; Guan, Qiang; Cheng, Feixiong

Allosteric drugs in biomolecular condensates: ways forward

生物分子凝聚体中的变构药物:前进之路

Nussinov, Ruth; Regev, Clil; Jang, Hyunbum

Oncogenic PI3Kα variants reveal graded conformational spectrum with mutation-specific cryptic pockets

致癌性PI3Kα变体揭示出具有突变特异性隐蔽口袋的梯度构象谱

Jang, Hyunbum; Yavuz, Bengi Ruken; Zhang, Mingzhen; Liu, Yonglan; Nussinov, Ruth

Cyclin-E/A/CDK1/2 Kinetic Landscapes Drive Cell Cycle Phase-Specific Progression and Guide Cyclin-E Degradation Strategy

细胞周期蛋白E/A/CDK1/2动力学图谱驱动细胞周期阶段特异性进程并指导细胞周期蛋白E降解策略

Zhang, Wengang; Bradburn, Devin; Liu, Yonglan; Jang, Hyunbum; Kõivomägi, Mardo; Nussinov, Ruth

Phosphorylation induces altered protonation states and allosterically regulates Rac1-RhoGDI complex

磷酸化作用诱导质子化状态改变,并变构调节 Rac1-RhoGDI 复合物。

Sinha, Krishnendu; Kumawat, Amit; Jang, Hyunbum; Nussinov, Ruth; Chakrabarty, Suman

The structural heterogeneity of AKT autoinhibition

AKT自身抑制的结构异质性

Xu, Liang; Eren, Meryem; Weako, Jackson; Jang, Hyunbum; Keskin, Ozlem; Gursoy, Attila; Nussinov, Ruth

Consensus on Human Epidermal Growth Factor Receptor 2 Overexpression Testing in Pan‐Tumor

关于泛肿瘤中人表皮生长因子受体2过表达检测的共识

Nussinov, Ruth; Wang, Zhe; Chen, Lin; Rao, Wei; Cao, Baoshan; Cai, Muyan; Fan, Xiangshan; Ji, Yuan; Li, Yuan; Song, Yan; Sun, Yan; Sun, Yu; Wu, Chunyan; Xia, Qingxin; Xi, Yanfeng; Xue, Liyan; Yin, Rutie; Liang, Han; Ying, Jianming

Allostery in Biomolecular Condensates

生物分子凝聚体中的变构

Nussinov, Ruth; Regev, Clil; Jang, Hyunbum

Repurposing AI for protein interactions and dynamics: opportunities, limitations, and lessons

将人工智能应用于蛋白质相互作用和动力学研究:机遇、局限性和经验教训

Ozdemir, E Sila; Jang, Hyunbum; Nussinov, Ruth; Gursoy, Attila; Keskin, Ozlem